Callyaerin G

Details

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Internal ID 3b32a339-65e5-4f42-aea5-6f2af83bb5ba
Taxonomy Organic Polymers > Polypeptides
IUPAC Name (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(3R,9S,15S,21S,23E,27S,30S)-21,27-bis(2-methylpropyl)-2,8,14,20,26,29-hexaoxo-1,7,13,19,22,25,28-heptazapentacyclo[28.3.0.03,7.09,13.015,19]tritriacont-23-ene-24-carbonyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid
SMILES (Canonical) CC(C)CC1C(=O)NC(=CNC(C(=O)N2CCCC2C(=O)N3CCCC3C(=O)N4CCCC4C(=O)N5CCCC5C(=O)N1)CC(C)C)C(=O)N6CCCC6C(=O)NC(CC7=CC=CC=C7)C(=O)NC(CC8=CC=CC=C8)C(=O)NC(CC9=CC=CC=C9)C(=O)O
SMILES (Isomeric) CC(C)C[C@H]1C(=O)N/C(=C/N[C@H](C(=O)N2CCC[C@H]2C(=O)N3CCC[C@H]3C(=O)N4CCC[C@@H]4C(=O)N5CCC[C@H]5C(=O)N1)CC(C)C)/C(=O)N6CCC[C@H]6C(=O)N[C@@H](CC7=CC=CC=C7)C(=O)N[C@@H](CC8=CC=CC=C8)C(=O)N[C@@H](CC9=CC=CC=C9)C(=O)O
InChI InChI=1S/C67H87N11O12/c1-41(2)35-46-57(79)73-51(40-68-49(36-42(3)4)62(84)76-32-16-27-54(76)65(87)78-34-18-29-56(78)66(88)77-33-17-28-55(77)64(86)75-31-15-26-53(75)61(83)70-46)63(85)74-30-14-25-52(74)60(82)71-48(38-44-21-10-6-11-22-44)58(80)69-47(37-43-19-8-5-9-20-43)59(81)72-50(67(89)90)39-45-23-12-7-13-24-45/h5-13,19-24,40-42,46-50,52-56,68H,14-18,25-39H2,1-4H3,(H,69,80)(H,70,83)(H,71,82)(H,72,81)(H,73,79)(H,89,90)/b51-40+/t46-,47-,48-,49-,50-,52-,53-,54-,55+,56-/m0/s1
InChI Key DYTFXINNOGEETQ-KUIQLQJMSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C67H87N11O12
Molecular Weight 1238.50 g/mol
Exact Mass 1237.65356725 g/mol
Topological Polar Surface Area (TPSA) 296.00 Ų
XlogP 6.30

Synonyms

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CHEMBL1253754

2D Structure

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2D Structure of Callyaerin G

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.92% 98.95%
CHEMBL3837 P07711 Cathepsin L 98.75% 96.61%
CHEMBL221 P23219 Cyclooxygenase-1 98.44% 90.17%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.14% 96.09%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 97.80% 98.33%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 97.73% 97.64%
CHEMBL333 P08253 Matrix metalloproteinase-2 96.90% 96.31%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 96.13% 98.24%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 96.02% 97.14%
CHEMBL3524 P56524 Histone deacetylase 4 95.17% 92.97%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.89% 95.56%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 92.15% 82.38%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 92.11% 94.45%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 91.99% 82.69%
CHEMBL2514 O95665 Neurotensin receptor 2 91.57% 100.00%
CHEMBL230 P35354 Cyclooxygenase-2 91.40% 89.63%
CHEMBL5103 Q969S8 Histone deacetylase 10 91.20% 90.08%
CHEMBL3310 Q96DB2 Histone deacetylase 11 90.80% 88.56%
CHEMBL1255126 O15151 Protein Mdm4 90.69% 90.20%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 90.62% 93.03%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 90.55% 93.00%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 90.32% 91.11%
CHEMBL4123 P30989 Neurotensin receptor 1 89.25% 96.67%
CHEMBL321 P14780 Matrix metalloproteinase 9 89.15% 92.12%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 88.51% 90.71%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.16% 95.89%
CHEMBL3137262 O60341 LSD1/CoREST complex 86.85% 97.09%
CHEMBL4198 P98170 Inhibitor of apoptosis protein 3 86.73% 97.79%
CHEMBL4588 P22894 Matrix metalloproteinase 8 86.21% 94.66%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 86.16% 95.00%
CHEMBL3359 P21462 Formyl peptide receptor 1 85.82% 93.56%
CHEMBL340 P08684 Cytochrome P450 3A4 85.26% 91.19%
CHEMBL5028 O14672 ADAM10 85.03% 97.50%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 83.75% 85.14%
CHEMBL4227 P25090 Lipoxin A4 receptor 83.66% 100.00%
CHEMBL4394 Q9NYA1 Sphingosine kinase 1 83.62% 96.03%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 81.44% 96.47%
CHEMBL332 P03956 Matrix metalloproteinase-1 81.32% 94.50%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 81.26% 91.81%
CHEMBL4208 P20618 Proteasome component C5 80.07% 90.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 52941213
LOTUS LTS0183057
wikiData Q104991561