AH-758

Details

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Internal ID 394ea94f-f2db-42a3-b6a2-f1a6a62f5baf
Taxonomy Phenylpropanoids and polyketides > Macrolides and analogues
IUPAC Name 4-O-[2-[3-hydroxy-4-[(4E,6E,12E,14Z)-10-hydroxy-3,15-dimethoxy-7,9,11,13-tetramethyl-16-oxo-1-oxacyclohexadeca-4,6,12,14-tetraen-2-yl]pentan-2-yl]-2-methoxy-5-methyl-6-propan-2-yloxan-4-yl] 1-O-[(2-oxo-1,3-dihydropyrrol-5-yl)methyl] (E)-but-2-enedioate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C45H67NO13/c1-25(2)42-30(7)36(57-39(49)19-18-38(48)56-24-33-16-17-37(47)46-33)23-45(55-12,59-42)32(9)41(51)31(8)43-34(53-10)15-13-14-26(3)20-28(5)40(50)29(6)21-27(4)22-35(54-11)44(52)58-43/h13-16,18-19,21-22,25,28-32,34,36,40-43,50-51H,17,20,23-24H2,1-12H3,(H,46,47)/b15-13+,19-18+,26-14+,27-21+,35-22-
InChI Key DHGOLDVSUHASSH-HFZALEEASA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C45H67NO13
Molecular Weight 830.00 g/mol
Exact Mass 829.46124119 g/mol
Topological Polar Surface Area (TPSA) 185.00 Ų
XlogP 5.90

Synonyms

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4-O-[2-[3-Hydroxy-4-[(4E,6E,12E,14Z)-10-hydroxy-3,15-dimethoxy-7,9,11,13-tetramethyl-16-oxo-1-oxacyclohexadeca-4,6,12,14-tetraen-2-yl]pentan-2-yl]-2-methoxy-5-methyl-6-propan-2-yloxan-4-yl] 1-O-[(2-oxo-1,3-dihydropyrrol-5-yl)methyl] (E)-but-2-enedioate

2D Structure

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2D Structure of AH-758

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 99.88% 85.14%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.25% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.66% 96.09%
CHEMBL253 P34972 Cannabinoid CB2 receptor 95.44% 97.25%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.63% 95.56%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 93.36% 94.45%
CHEMBL2581 P07339 Cathepsin D 92.58% 98.95%
CHEMBL3137262 O60341 LSD1/CoREST complex 92.08% 97.09%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 92.07% 91.07%
CHEMBL1293249 Q13887 Kruppel-like factor 5 91.34% 86.33%
CHEMBL2535 P11166 Glucose transporter 91.13% 98.75%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 90.46% 96.95%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 90.15% 96.77%
CHEMBL4657 Q6V1X1 Dipeptidyl peptidase VIII 89.91% 97.21%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 88.24% 99.23%
CHEMBL3359 P21462 Formyl peptide receptor 1 87.86% 93.56%
CHEMBL3401 O75469 Pregnane X receptor 87.48% 94.73%
CHEMBL1806 P11388 DNA topoisomerase II alpha 86.56% 89.00%
CHEMBL4481 P35228 Nitric oxide synthase, inducible 86.35% 94.80%
CHEMBL5608 Q16288 NT-3 growth factor receptor 85.34% 95.89%
CHEMBL340 P08684 Cytochrome P450 3A4 82.25% 91.19%
CHEMBL1902 P62942 FK506-binding protein 1A 82.18% 97.05%
CHEMBL4208 P20618 Proteasome component C5 81.49% 90.00%
CHEMBL218 P21554 Cannabinoid CB1 receptor 81.10% 96.61%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 80.86% 95.89%
CHEMBL3060 Q9Y345 Glycine transporter 2 80.28% 99.17%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 10463186
LOTUS LTS0238907
wikiData Q77521721