Benadrostin

Details

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Internal ID d32f8d5a-7770-4789-a83d-f13fc02482a2
Taxonomy Organoheterocyclic compounds > Benzoxazines
IUPAC Name 8-hydroxy-1,3-benzoxazine-2,4-dione
SMILES (Canonical) C1=CC2=C(C(=C1)O)OC(=O)NC2=O
SMILES (Isomeric) C1=CC2=C(C(=C1)O)OC(=O)NC2=O
InChI InChI=1S/C8H5NO4/c10-5-3-1-2-4-6(5)13-8(12)9-7(4)11/h1-3,10H,(H,9,11,12)
InChI Key BQIRLGRTNUTGAT-UHFFFAOYSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C8H5NO4
Molecular Weight 179.13 g/mol
Exact Mass 179.02185764 g/mol
Topological Polar Surface Area (TPSA) 75.60 Ų
XlogP 0.70

Synonyms

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117241-60-8
8-hydroxy-1,3-benzoxazine-2,4-dione
8-Hydroxy-2H-1,3-benzoxazine-2,4(3H)-dione
2H-1,3-Benzoxazine-2,4(3H)-dione, 8-hydroxy-
SCHEMBL16431150
DTXSID00151728
AKOS006273706
8-hydroxy-2H-1,3-benzoxazine-2,4-dione

2D Structure

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2D Structure of Benadrostin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 95.49% 91.11%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 94.75% 99.23%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.23% 95.56%
CHEMBL3401 O75469 Pregnane X receptor 89.08% 94.73%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 88.15% 94.45%
CHEMBL1806 P11388 DNA topoisomerase II alpha 87.95% 89.00%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 87.53% 94.00%
CHEMBL2581 P07339 Cathepsin D 87.24% 98.95%
CHEMBL3192 Q9BY41 Histone deacetylase 8 86.69% 93.99%
CHEMBL2535 P11166 Glucose transporter 84.68% 98.75%
CHEMBL1937 Q92769 Histone deacetylase 2 84.66% 94.75%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 83.87% 99.15%
CHEMBL3830 Q2M2I8 Adaptor-associated kinase 83.80% 83.10%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 197266
LOTUS LTS0135637
wikiData Q104907948