Bacillcoumacin G

Details

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Internal ID addabc55-dd29-42d8-af59-6a0ee987372d
Taxonomy Organoheterocyclic compounds > Benzopyrans > 2-benzopyrans
IUPAC Name (2Z)-N-[(1S)-1-[(3S)-8-hydroxy-1-oxo-3,4-dihydroisochromen-3-yl]-3-methylbutyl]-2-(5-oxopyrrolidin-2-ylidene)acetamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C20H24N2O5/c1-11(2)8-14(22-18(25)10-13-6-7-17(24)21-13)16-9-12-4-3-5-15(23)19(12)20(26)27-16/h3-5,10-11,14,16,23H,6-9H2,1-2H3,(H,21,24)(H,22,25)/b13-10-/t14-,16-/m0/s1
InChI Key JXGHXIFIIWVALX-JJPUIBJASA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C20H24N2O5
Molecular Weight 372.40 g/mol
Exact Mass 372.16852187 g/mol
Topological Polar Surface Area (TPSA) 105.00 Ų
XlogP 2.50

Synonyms

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(3Z)-N-((1S)-1-((3S)-8-hydroxy-1-oxo-3,4-dihydroisochromen-3-yl)-3-methylbutyl)-3-(5-oxopyrrolidin-3-ylidene)propanamide
(3Z)-N-[(1S)-1-[(3S)-8-hydroxy-1-oxo-3,4-dihydroisochromen-3-yl]-3-methylbutyl]-3-(5-oxopyrrolidin-3-ylidene)propanamide
RefChem:116231
CHEBI:198308
(2Z)-N-[(1S)-1-[(3S)-8-hydroxy-1-oxo-3,4-dihydroisochromen-3-yl]-3-methylbutyl]-2-(5-oxopyrrolidin-2-ylidene)acetamide

2D Structure

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2D Structure of Bacillcoumacin G

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.81% 91.11%
CHEMBL2581 P07339 Cathepsin D 98.47% 98.95%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 97.48% 94.45%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 95.97% 96.09%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.61% 95.56%
CHEMBL3830 Q2M2I8 Adaptor-associated kinase 93.43% 83.10%
CHEMBL1937 Q92769 Histone deacetylase 2 93.17% 94.75%
CHEMBL3359 P21462 Formyl peptide receptor 1 91.59% 93.56%
CHEMBL3192 Q9BY41 Histone deacetylase 8 91.48% 93.99%
CHEMBL1806 P11388 DNA topoisomerase II alpha 88.81% 89.00%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 88.56% 99.23%
CHEMBL2553 Q15418 Ribosomal protein S6 kinase alpha 1 88.15% 85.11%
CHEMBL3137262 O60341 LSD1/CoREST complex 87.25% 97.09%
CHEMBL2964 P36507 Dual specificity mitogen-activated protein kinase kinase 2 86.72% 80.00%
CHEMBL5608 Q16288 NT-3 growth factor receptor 84.20% 95.89%
CHEMBL1994 P08235 Mineralocorticoid receptor 83.78% 100.00%
CHEMBL5028 O14672 ADAM10 83.40% 97.50%
CHEMBL3401 O75469 Pregnane X receptor 83.33% 94.73%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 82.59% 90.71%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 82.32% 99.15%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 81.68% 96.38%
CHEMBL221 P23219 Cyclooxygenase-1 81.60% 90.17%
CHEMBL4227 P25090 Lipoxin A4 receptor 81.06% 100.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 80.97% 93.03%
CHEMBL2535 P11166 Glucose transporter 80.62% 98.75%
CHEMBL5103 Q969S8 Histone deacetylase 10 80.46% 90.08%
CHEMBL236 P41143 Delta opioid receptor 80.33% 99.35%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139583338
LOTUS LTS0089206
wikiData Q75059205