Aspergillicin A

Details

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Internal ID d258b12d-4653-4eb8-8a75-7ff08183422e
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name N-[(3S,9R,12S,13R,16S,19S,22S)-9-[(2S)-butan-2-yl]-19-[(4-methoxyphenyl)methyl]-13,20-dimethyl-2,8,11,15,18,21-hexaoxo-16-propan-2-yl-14-oxa-1,7,10,17,20-pentazatricyclo[20.3.0.03,7]pentacosan-12-yl]acetamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C38H56N6O9/c1-9-22(4)31-37(50)44-19-11-13-28(44)36(49)43-18-10-12-27(43)35(48)42(7)29(20-25-14-16-26(52-8)17-15-25)33(46)40-30(21(2)3)38(51)53-23(5)32(34(47)41-31)39-24(6)45/h14-17,21-23,27-32H,9-13,18-20H2,1-8H3,(H,39,45)(H,40,46)(H,41,47)/t22-,23+,27-,28-,29-,30-,31+,32-/m0/s1
InChI Key NCCHYDXMXHIKMK-FVOMNUFISA-N
Popularity 4 references in papers

Physical and Chemical Properties

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Molecular Formula C38H56N6O9
Molecular Weight 740.90 g/mol
Exact Mass 740.41087739 g/mol
Topological Polar Surface Area (TPSA) 184.00 Ų
XlogP 3.10

Synonyms

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N-[(3S,9R,12S,13R,16S,19S,22S)-9-[(2S)-butan-2-yl]-19-[(4-methoxyphenyl)methyl]-13,20-dimethyl-2,8,11,15,18,21-hexaoxo-16-propan-2-yl-14-oxa-1,7,10,17,20-pentazatricyclo[20.3.0.03,7]pentacosan-12-yl]acetamide
N-((3S,9R,12S,13R,16S,19S,22S)-9-((2S)-Butan-2-yl)-11,18-dihydroxy-19-((4-methoxyphenyl)methyl)-13,20-dimethyl-2,8,15,21-tetraoxo-16-(propan-2-yl)-14-oxa-1,7,10,17,20-pentaazatricyclo(20.3.0.0,)pentacosa-10,17-dien-12-yl)ethanimidate
N-((3S,9R,12S,13R,16S,19S,22S)-9-((2S)-butan-2-yl)-19-((4-methoxyphenyl)methyl)-13,20-dimethyl-2,8,11,15,18,21-hexaoxo-16-propan-2-yl-14-oxa-1,7,10,17,20-pentazatricyclo(20.3.0.03,7)pentacosan-12-yl)acetamide
N-[(3S,9R,12S,13R,16S,19S,22S)-9-[(2S)-Butan-2-yl]-11,18-dihydroxy-19-[(4-methoxyphenyl)methyl]-13,20-dimethyl-2,8,15,21-tetraoxo-16-(propan-2-yl)-14-oxa-1,7,10,17,20-pentaazatricyclo[20.3.0.0,]pentacosa-10,17-dien-12-yl]ethanimidate
RefChem:114812
SCHEMBL1592839
CHEMBL5082301
CHEBI:212622

2D Structure

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2D Structure of Aspergillicin A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.62% 98.95%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 99.45% 85.14%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.30% 96.09%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.94% 94.45%
CHEMBL3837 P07711 Cathepsin L 94.16% 96.61%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.89% 95.56%
CHEMBL5608 Q16288 NT-3 growth factor receptor 93.61% 95.89%
CHEMBL4208 P20618 Proteasome component C5 93.44% 90.00%
CHEMBL333 P08253 Matrix metalloproteinase-2 92.66% 96.31%
CHEMBL4588 P22894 Matrix metalloproteinase 8 92.32% 94.66%
CHEMBL255 P29275 Adenosine A2b receptor 92.08% 98.59%
CHEMBL5103 Q969S8 Histone deacetylase 10 92.03% 90.08%
CHEMBL253 P34972 Cannabinoid CB2 receptor 91.40% 97.25%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 91.29% 91.11%
CHEMBL3060 Q9Y345 Glycine transporter 2 90.07% 99.17%
CHEMBL3137262 O60341 LSD1/CoREST complex 88.85% 97.09%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 88.69% 94.00%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 87.13% 93.00%
CHEMBL4072 P07858 Cathepsin B 86.17% 93.67%
CHEMBL1902 P62942 FK506-binding protein 1A 84.45% 97.05%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 84.41% 95.89%
CHEMBL226 P30542 Adenosine A1 receptor 84.17% 95.93%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 83.31% 90.71%
CHEMBL1293249 Q13887 Kruppel-like factor 5 83.10% 86.33%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 81.81% 94.33%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 81.71% 97.14%
CHEMBL2443 P49862 Kallikrein 7 81.50% 94.00%
CHEMBL4531 P17931 Galectin-3 81.07% 96.90%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 10930650
LOTUS LTS0120212
wikiData Q77494660