Acyclolaxaphycin A

Details

Top
Internal ID c68efc2c-43a9-417f-9ddf-cf9644988102
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides
IUPAC Name 2-[[(2S)-2-[[(2R,3S)-2-[[(2S,3S)-2-[[(2R)-2-[[(2R)-2-[[(2S)-2-[[(2S,4R)-1-[(E)-2-[[(2S)-2-[[(3R)-3-aminooctanoyl]amino]-4-hydroxybutanoyl]amino]but-2-enoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-4-hydroxybutanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-methylpentanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoyl]amino]acetic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C60H99N11O15/c1-11-15-17-22-39(61)30-48(75)63-42(23-25-72)53(79)64-41(14-4)60(86)71-33-40(74)31-47(71)57(83)65-43(24-26-73)54(80)67-46(29-38-20-18-16-19-21-38)55(81)66-45(28-35(7)8)56(82)69-51(37(10)13-3)59(85)70-50(36(9)12-2)58(84)68-44(27-34(5)6)52(78)62-32-49(76)77/h14,16,18-21,34-37,39-40,42-47,50-51,72-74H,11-13,15,17,22-33,61H2,1-10H3,(H,62,78)(H,63,75)(H,64,79)(H,65,83)(H,66,81)(H,67,80)(H,68,84)(H,69,82)(H,70,85)(H,76,77)/b41-14+/t36-,37-,39+,40+,42-,43-,44-,45+,46+,47-,50+,51-/m0/s1
InChI Key WSDZDIHEDAEEBI-NZVCJXAPSA-N
Popularity 3 references in papers

Physical and Chemical Properties

Top
Molecular Formula C60H99N11O15
Molecular Weight 1214.50 g/mol
Exact Mass 1213.73221149 g/mol
Topological Polar Surface Area (TPSA) 406.00 Ų
XlogP 1.20

Synonyms

Top
There are no found synonyms.

2D Structure

Top
2D Structure of Acyclolaxaphycin A

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.98% 98.95%
CHEMBL3837 P07711 Cathepsin L 99.36% 96.61%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.49% 96.09%
CHEMBL4801 P29466 Caspase-1 97.91% 96.85%
CHEMBL221 P23219 Cyclooxygenase-1 97.71% 90.17%
CHEMBL3060 Q9Y345 Glycine transporter 2 97.56% 99.17%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 97.49% 98.33%
CHEMBL4657 Q6V1X1 Dipeptidyl peptidase VIII 97.01% 97.21%
CHEMBL2514 O95665 Neurotensin receptor 2 96.80% 100.00%
CHEMBL3359 P21462 Formyl peptide receptor 1 96.53% 93.56%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 95.91% 96.95%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.68% 95.56%
CHEMBL230 P35354 Cyclooxygenase-2 95.44% 89.63%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 95.25% 97.64%
CHEMBL340 P08684 Cytochrome P450 3A4 95.11% 91.19%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 94.55% 97.23%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.47% 91.11%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 93.68% 97.14%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 93.39% 91.81%
CHEMBL1907591 P30926 Neuronal acetylcholine receptor; alpha4/beta4 93.32% 100.00%
CHEMBL3137262 O60341 LSD1/CoREST complex 92.05% 97.09%
CHEMBL4769 O95749 Geranylgeranyl pyrophosphate synthetase 91.82% 92.08%
CHEMBL3891 P07384 Calpain 1 91.23% 93.04%
CHEMBL4123 P30989 Neurotensin receptor 1 90.74% 96.67%
CHEMBL5701 Q9H2K8 Serine/threonine-protein kinase TAO3 90.36% 96.67%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 89.25% 82.69%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 88.65% 93.00%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 88.08% 90.71%
CHEMBL4227 P25090 Lipoxin A4 receptor 87.81% 100.00%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 87.35% 96.47%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 87.27% 96.00%
CHEMBL1255126 O15151 Protein Mdm4 87.07% 90.20%
CHEMBL4462 Q8IXJ6 NAD-dependent deacetylase sirtuin 2 86.41% 90.24%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 86.16% 88.42%
CHEMBL1944495 P28065 Proteasome subunit beta type-9 86.09% 97.50%
CHEMBL5939 Q9NZ08 Endoplasmic reticulum aminopeptidase 1 84.88% 100.00%
CHEMBL2288 Q13526 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 84.80% 91.71%
CHEMBL237 P41145 Kappa opioid receptor 84.76% 98.10%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 84.49% 95.89%
CHEMBL5261 Q7L7X3 Serine/threonine-protein kinase TAO1 84.15% 89.33%
CHEMBL5028 O14672 ADAM10 84.01% 97.50%
CHEMBL3004 P33527 Multidrug resistance-associated protein 1 82.45% 96.37%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 81.79% 96.90%
CHEMBL2885 P07451 Carbonic anhydrase III 81.66% 87.45%
CHEMBL1781 P11387 DNA topoisomerase I 81.06% 97.00%
CHEMBL1821 P08173 Muscarinic acetylcholine receptor M4 81.00% 94.08%
CHEMBL4506 Q96EB6 NAD-dependent deacetylase sirtuin 1 80.97% 88.33%
CHEMBL216 P11229 Muscarinic acetylcholine receptor M1 80.85% 94.23%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 80.61% 95.00%
CHEMBL3892 Q99500 Sphingosine 1-phosphate receptor Edg-3 80.22% 97.29%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 146682308
LOTUS LTS0098323
wikiData Q105311800