Acetyltylophoroside

Details

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Internal ID 449759af-d59e-459f-ac5c-4cd1d8305480
Taxonomy Lipids and lipid-like molecules > Steroids and steroid derivatives > Oxosteroids > 16-oxosteroids
IUPAC Name [(1R,2R,4aS,4bR,8R,8aS,9S,10aR)-1,8-diacetyloxy-7-[(2S,4S,5R,6S)-5-[(2S,3R,4R,5R,6S)-3-acetyloxy-4-methoxy-6-methyl-5-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]oxy-4-methoxy-6-methyloxan-2-yl]oxy-2-[(2S)-2-methoxy-2-methyl-5-oxofuran-3-yl]-2,4b-dimethyl-1,3,4,4a,5,8,8a,9,10,10a-decahydrophenanthren-9-yl] acetate
SMILES (Canonical) CC1C(C(CC(O1)OC2=CCC3(C4CCC(C(C4CC(C3C2OC(=O)C)OC(=O)C)OC(=O)C)(C)C5=CC(=O)OC5(C)OC)C)OC)OC6C(C(C(C(O6)C)OC7C(C(C(C(O7)CO)O)O)O)OC)OC(=O)C
SMILES (Isomeric) C[C@H]1[C@H]([C@H](C[C@@H](O1)OC2=CC[C@@]3([C@H]4CC[C@]([C@@H]([C@@H]4C[C@@H]([C@H]3[C@H]2OC(=O)C)OC(=O)C)OC(=O)C)(C)C5=CC(=O)O[C@]5(C)OC)C)OC)O[C@H]6[C@@H]([C@@H]([C@@H]([C@@H](O6)C)O[C@H]7[C@@H]([C@H]([C@@H]([C@H](O7)CO)O)O)O)OC)OC(=O)C
InChI InChI=1S/C50H74O23/c1-21-40(71-47-44(67-25(5)54)43(61-11)41(22(2)64-47)72-46-39(59)38(58)37(57)32(20-51)70-46)31(60-10)18-35(63-21)69-29-14-16-48(7)28-13-15-49(8,33-19-34(56)73-50(33,9)62-12)45(68-26(6)55)27(28)17-30(65-23(3)52)36(48)42(29)66-24(4)53/h14,19,21-22,27-28,30-32,35-47,51,57-59H,13,15-18,20H2,1-12H3/t21-,22-,27+,28-,30-,31-,32+,35-,36-,37+,38-,39+,40+,41+,42-,43+,44+,45+,46-,47-,48+,49+,50-/m0/s1
InChI Key FSCPZINTFYRQQD-SDGPZJJRSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C50H74O23
Molecular Weight 1043.10 g/mol
Exact Mass 1042.46208860 g/mol
Topological Polar Surface Area (TPSA) 296.00 Ų
XlogP 1.30

Synonyms

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135247-54-0
[(1R,2R,4aS,4bR,8R,8aS,9S,10aR)-1,8-diacetyloxy-7-[(2S,4S,5R,6S)-5-[(2S,3R,4R,5R,6S)-3-acetyloxy-4-methoxy-6-methyl-5-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyoxan-2-yl]oxy-4-methoxy-6-methyloxan-2-yl]oxy-2-[(2S)-2-methoxy-2-methyl-5-oxofuran-3-yl]-2,4b-dimethyl-1,3,4,4a,5,8,8a,9,10,10a-decahydrophenanthren-9-yl] acetate
((1R,2R,4aS,4bR,8R,8aS,9S,10aR)-1,8-diacetyloxy-7-((2S,4S,5R,6S)-5-((2S,3R,4R,5R,6S)-3-acetyloxy-4-methoxy-6-methyl-5-((2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl)oxyoxan-2-yl)oxy-4-methoxy-6-methyloxan-2-yl)oxy-2-((2S)-2-methoxy-2-methyl-5-oxofuran-3-yl)-2,4b-dimethyl-1,3,4,4a,5,8,8a,9,10,10a-decahydrophenanthren-9-yl) acetate
RefChem:109208
5-Methoxy-5-methyl-4-(1,8,9-tris(acetyloxy)-7-((O-beta-D-glucopyranosyl)-(1-4)-O-2-O-acetyl-6-deoxy-3-O-methyl-alpha-L-talopyranosyl-(1-4)-2,6-dideoxy-3-O-methyl-alpha-L-lyxo-hexopyranosyl)oxy)-1,2,3,4,4a,4b,5,8,8a,9,10,10a-2(5H)-furanone
2(5H)-Furanone, 5-methoxy-5-methyl-4-(1,8,9-tris(acetyloxy)-7-((O-beta-D-glucopyranosyl)-(1-4)-O-2-O-acetyl-6-deoxy-3-O-methyl-alpha-L-talopyranosyl-(1-4)-2,6-dideoxy-3-O-methyl-alpha-L-lyxo-hexopyranosyl)oxy)-1,2,3,4,4a,4b,5,8,8a,9,10,10a-

2D Structure

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2D Structure of Acetyltylophoroside

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.42% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.68% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 96.55% 85.14%
CHEMBL2581 P07339 Cathepsin D 95.45% 98.95%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 94.25% 96.77%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 92.58% 95.89%
CHEMBL3137262 O60341 LSD1/CoREST complex 92.49% 97.09%
CHEMBL1994 P08235 Mineralocorticoid receptor 91.20% 100.00%
CHEMBL253 P34972 Cannabinoid CB2 receptor 90.43% 97.25%
CHEMBL1293249 Q13887 Kruppel-like factor 5 90.14% 86.33%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 90.08% 94.45%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 89.76% 94.00%
CHEMBL5255 O00206 Toll-like receptor 4 89.52% 92.50%
CHEMBL226 P30542 Adenosine A1 receptor 89.29% 95.93%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.26% 89.00%
CHEMBL3714130 P46095 G-protein coupled receptor 6 88.91% 97.36%
CHEMBL340 P08684 Cytochrome P450 3A4 87.30% 91.19%
CHEMBL5608 Q16288 NT-3 growth factor receptor 87.25% 95.89%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 86.96% 97.33%
CHEMBL241 Q14432 Phosphodiesterase 3A 86.63% 92.94%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 86.48% 95.56%
CHEMBL1871 P10275 Androgen Receptor 85.57% 96.43%
CHEMBL1293277 O15118 Niemann-Pick C1 protein 83.75% 81.11%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 83.69% 99.23%
CHEMBL4481 P35228 Nitric oxide synthase, inducible 83.47% 94.80%
CHEMBL204 P00734 Thrombin 82.25% 96.01%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 81.72% 97.14%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 80.95% 94.33%
CHEMBL5028 O14672 ADAM10 80.56% 97.50%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 3086643
LOTUS LTS0103007
wikiData Q105000580