Destruxin A

Details

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Internal ID 40d714b6-43a6-4ca8-b5a6-f44617bdbdae
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (3R,10S,13S,16S,19S)-16-[(2S)-butan-2-yl]-10,11,14-trimethyl-13-propan-2-yl-3-prop-2-enyl-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone
SMILES (Canonical) CCC(C)C1C(=O)N(C(C(=O)N(C(C(=O)NCCC(=O)OC(C(=O)N2CCCC2C(=O)N1)CC=C)C)C)C(C)C)C
SMILES (Isomeric) CC[C@H](C)[C@H]1C(=O)N([C@H](C(=O)N([C@H](C(=O)NCCC(=O)O[C@@H](C(=O)N2CCC[C@H]2C(=O)N1)CC=C)C)C)C(C)C)C
InChI InChI=1S/C29H47N5O7/c1-9-12-21-27(38)34-16-11-13-20(34)26(37)31-23(18(5)10-2)28(39)33(8)24(17(3)4)29(40)32(7)19(6)25(36)30-15-14-22(35)41-21/h9,17-21,23-24H,1,10-16H2,2-8H3,(H,30,36)(H,31,37)/t18-,19-,20-,21+,23-,24-/m0/s1
InChI Key XIYSEKITPHTMJT-OCCJOITDSA-N
Popularity 39 references in papers

Physical and Chemical Properties

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Molecular Formula C29H47N5O7
Molecular Weight 577.70 g/mol
Exact Mass 577.34754886 g/mol
Topological Polar Surface Area (TPSA) 145.00 Ų
XlogP 2.30

Synonyms

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6686-70-0
255H1K2LFG
(3R,10S,13S,16S,19S)-16-[(2S)-butan-2-yl]-10,11,14-trimethyl-13-propan-2-yl-3-prop-2-enyl-4-oxa-1,8,11,14,17-pentazabicyclo[17.3.0]docosane-2,5,9,12,15,18-hexone
UNII-255H1K2LFG
NSC-361126
Destruxin A from Metarrhizium anisopliae
NSC 361126
DESTRUXIN DA
BRN 0601694
CHEMBL4524055
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of Destruxin A

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 98.93% 98.95%
CHEMBL253 P34972 Cannabinoid CB2 receptor 98.49% 97.25%
CHEMBL333 P08253 Matrix metalloproteinase-2 98.00% 96.31%
CHEMBL4588 P22894 Matrix metalloproteinase 8 97.69% 94.66%
CHEMBL5103 Q969S8 Histone deacetylase 10 97.56% 90.08%
CHEMBL1902 P62942 FK506-binding protein 1A 95.33% 97.05%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 94.53% 96.09%
CHEMBL1937 Q92769 Histone deacetylase 2 94.21% 94.75%
CHEMBL3524 P56524 Histone deacetylase 4 93.24% 92.97%
CHEMBL321 P14780 Matrix metalloproteinase 9 92.54% 92.12%
CHEMBL228 P31645 Serotonin transporter 92.29% 95.51%
CHEMBL332 P03956 Matrix metalloproteinase-1 92.10% 94.50%
CHEMBL3137262 O60341 LSD1/CoREST complex 91.60% 97.09%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 90.96% 82.38%
CHEMBL2996 Q05655 Protein kinase C delta 90.89% 97.79%
CHEMBL5608 Q16288 NT-3 growth factor receptor 90.65% 95.89%
CHEMBL2189110 Q15910 Histone-lysine N-methyltransferase EZH2 90.25% 97.50%
CHEMBL255 P29275 Adenosine A2b receptor 90.05% 98.59%
CHEMBL299 P17252 Protein kinase C alpha 89.72% 98.03%
CHEMBL5203 P33316 dUTP pyrophosphatase 89.71% 99.18%
CHEMBL325 Q13547 Histone deacetylase 1 89.47% 95.92%
CHEMBL4616 Q92847 Ghrelin receptor 87.92% 92.00%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 87.78% 93.40%
CHEMBL3837 P07711 Cathepsin L 87.76% 96.61%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 87.45% 95.56%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 87.38% 93.00%
CHEMBL226 P30542 Adenosine A1 receptor 87.12% 95.93%
CHEMBL1806 P11388 DNA topoisomerase II alpha 86.36% 89.00%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 85.92% 91.03%
CHEMBL217 P14416 Dopamine D2 receptor 85.87% 95.62%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 85.71% 90.24%
CHEMBL4005 P42336 PI3-kinase p110-alpha subunit 85.57% 97.47%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 85.54% 90.71%
CHEMBL3310 Q96DB2 Histone deacetylase 11 85.11% 88.56%
CHEMBL2443 P49862 Kallikrein 7 83.73% 94.00%
CHEMBL1949 P62937 Cyclophilin A 83.45% 98.57%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 83.19% 94.45%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 83.03% 96.47%
CHEMBL4835 P00338 L-lactate dehydrogenase A chain 82.62% 95.34%
CHEMBL3691 Q13822 Autotaxin 82.61% 96.39%
CHEMBL1994 P08235 Mineralocorticoid receptor 82.38% 100.00%
CHEMBL4208 P20618 Proteasome component C5 80.98% 90.00%
CHEMBL1293249 Q13887 Kruppel-like factor 5 80.78% 86.33%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 11421831
LOTUS LTS0136046
wikiData Q27253912