Tsushimycin

Details

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Internal ID 9e2c4f96-06ab-4720-863d-cb5384372aeb
Taxonomy Organic acids and derivatives > Peptidomimetics > Hybrid peptides
IUPAC Name (3S)-4-[[(3S,7S,13S,16S,23S,29S,35S)-16-[(1R)-1-aminoethyl]-32-(1-carboxyethyl)-23,29-bis(carboxymethyl)-4-methyl-2,6,12,15,18,20,22,25,28,31,34-undecaoxo-13-propan-2-yl-1,5,11,14,17,21,24,27,30,33-decazatricyclo[33.4.0.07,11]nonatriacontan-3-yl]amino]-3-[[(E)-12-methyltridec-3-enoyl]amino]-4-oxobutanoic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C60H93N13O21/c1-30(2)19-14-12-10-8-9-11-13-15-22-40(74)64-37(27-46(82)83)53(86)71-50-34(7)63-54(87)39-21-18-24-73(39)58(91)47(31(3)4)69-57(90)49(33(6)61)67-41(75)28-42(76)68-52(85)36(26-45(80)81)65-43(77)29-62-51(84)35(25-44(78)79)66-56(89)48(32(5)60(93)94)70-55(88)38-20-16-17-23-72(38)59(50)92/h13,15,30-39,47-50H,8-12,14,16-29,61H2,1-7H3,(H,62,84)(H,63,87)(H,64,74)(H,65,77)(H,66,89)(H,67,75)(H,69,90)(H,70,88)(H,71,86)(H,78,79)(H,80,81)(H,82,83)(H,93,94)(H,68,76,85)/b15-13+/t32?,33-,34?,35+,36+,37+,38+,39+,47+,48?,49+,50+/m1/s1
InChI Key UYDPPDOTOCWOBT-DIKMMNQVSA-N
Popularity 8 references in papers

Physical and Chemical Properties

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Molecular Formula C60H93N13O21
Molecular Weight 1332.50 g/mol
Exact Mass 1331.66089703 g/mol
Topological Polar Surface Area (TPSA) 524.00 Ų
XlogP -2.50

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of Tsushimycin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.74% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.53% 96.09%
CHEMBL236 P41143 Delta opioid receptor 99.36% 99.35%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.31% 91.11%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 98.10% 91.03%
CHEMBL4801 P29466 Caspase-1 98.05% 96.85%
CHEMBL3524 P56524 Histone deacetylase 4 96.99% 92.97%
CHEMBL226 P30542 Adenosine A1 receptor 96.84% 95.93%
CHEMBL221 P23219 Cyclooxygenase-1 96.60% 90.17%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 96.33% 93.00%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 95.42% 96.11%
CHEMBL5103 Q969S8 Histone deacetylase 10 94.96% 90.08%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 94.89% 82.38%
CHEMBL3060 Q9Y345 Glycine transporter 2 94.79% 99.17%
CHEMBL1902 P62942 FK506-binding protein 1A 94.46% 97.05%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 94.36% 95.50%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 94.22% 90.71%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 93.25% 94.45%
CHEMBL4588 P22894 Matrix metalloproteinase 8 93.19% 94.66%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 92.48% 98.33%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 92.00% 96.90%
CHEMBL4071 P08311 Cathepsin G 91.69% 94.64%
CHEMBL5203 P33316 dUTP pyrophosphatase 91.61% 99.18%
CHEMBL5608 Q16288 NT-3 growth factor receptor 90.11% 95.89%
CHEMBL3468 P55210 Caspase-7 88.52% 95.68%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 88.36% 93.03%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 88.34% 96.38%
CHEMBL4979 P13866 Sodium/glucose cotransporter 1 88.29% 98.24%
CHEMBL3359 P21462 Formyl peptide receptor 1 88.10% 93.56%
CHEMBL2094135 Q96BI3 Gamma-secretase 87.99% 98.05%
CHEMBL2781 P19634 Sodium/hydrogen exchanger 1 87.84% 90.24%
CHEMBL3137262 O60341 LSD1/CoREST complex 87.58% 97.09%
CHEMBL2413 P32246 C-C chemokine receptor type 1 87.52% 89.50%
CHEMBL333 P08253 Matrix metalloproteinase-2 86.92% 96.31%
CHEMBL2514 O95665 Neurotensin receptor 2 86.32% 100.00%
CHEMBL2001 Q9H244 Purinergic receptor P2Y12 85.85% 96.00%
CHEMBL5966 P55899 IgG receptor FcRn large subunit p51 85.76% 90.93%
CHEMBL4394 Q9NYA1 Sphingosine kinase 1 85.65% 96.03%
CHEMBL1937 Q92769 Histone deacetylase 2 85.38% 94.75%
CHEMBL2443 P49862 Kallikrein 7 85.16% 94.00%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 84.78% 97.64%
CHEMBL1806 P11388 DNA topoisomerase II alpha 84.78% 89.00%
CHEMBL325 Q13547 Histone deacetylase 1 84.45% 95.92%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 83.89% 96.47%
CHEMBL340 P08684 Cytochrome P450 3A4 83.74% 91.19%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 83.42% 95.56%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 82.93% 82.69%
CHEMBL5255 O00206 Toll-like receptor 4 81.89% 92.50%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 81.72% 94.33%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 81.52% 97.14%
CHEMBL3784 Q09472 Histone acetyltransferase p300 81.01% 93.33%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 80.97% 88.42%
CHEMBL4618 P09960 Leukotriene A4 hydrolase 80.46% 97.86%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139589218
LOTUS LTS0133162
wikiData Q105281325