Duocarmycin C1

Details

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Internal ID d464dfd4-f2d1-4886-8e97-0607dec9de27
Taxonomy Organoheterocyclic compounds > Quinolines and derivatives > Pyrroloquinolines
IUPAC Name methyl 8-chloro-4-hydroxy-2-methyl-1-oxo-6-(5,6,7-trimethoxy-1H-indole-2-carbonyl)-3,7,8,9-tetrahydropyrrolo[3,2-f]quinoline-2-carboxylate
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C26H26ClN3O8/c1-26(25(34)38-5)23(32)18-13-8-12(27)10-30(15(13)9-16(31)20(18)29-26)24(33)14-6-11-7-17(35-2)21(36-3)22(37-4)19(11)28-14/h6-7,9,12,28-29,31H,8,10H2,1-5H3
InChI Key ILRQRCTVPANBBE-UHFFFAOYSA-N
Popularity 10 references in papers

Physical and Chemical Properties

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Molecular Formula C26H26ClN3O8
Molecular Weight 544.00 g/mol
Exact Mass 543.1408425 g/mol
Topological Polar Surface Area (TPSA) 139.00 Ų
XlogP 3.50

Synonyms

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methyl 8-chloro-4-hydroxy-2-methyl-1-oxo-6-(5,6,7-trimethoxy-1H-indole-2-carbonyl)-3,7,8,9-tetrahydropyrrolo[3,2-f]quinoline-2-carboxylate

2D Structure

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2D Structure of Duocarmycin C1

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.57% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.39% 96.09%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 98.21% 94.45%
CHEMBL4040 P28482 MAP kinase ERK2 96.67% 83.82%
CHEMBL261 P00915 Carbonic anhydrase I 94.94% 96.76%
CHEMBL4302 P08183 P-glycoprotein 1 94.48% 92.98%
CHEMBL2535 P11166 Glucose transporter 94.31% 98.75%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.16% 95.56%
CHEMBL340 P08684 Cytochrome P450 3A4 92.70% 91.19%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 92.62% 85.14%
CHEMBL2581 P07339 Cathepsin D 91.89% 98.95%
CHEMBL1293249 Q13887 Kruppel-like factor 5 90.47% 86.33%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 88.97% 91.03%
CHEMBL3060 Q9Y345 Glycine transporter 2 88.15% 99.17%
CHEMBL4208 P20618 Proteasome component C5 88.10% 90.00%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 87.87% 93.03%
CHEMBL1937 Q92769 Histone deacetylase 2 87.76% 94.75%
CHEMBL3137262 O60341 LSD1/CoREST complex 87.39% 97.09%
CHEMBL230 P35354 Cyclooxygenase-2 86.94% 89.63%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 86.84% 93.40%
CHEMBL205 P00918 Carbonic anhydrase II 84.99% 98.44%
CHEMBL3788 O00444 Serine/threonine-protein kinase PLK4 84.69% 83.65%
CHEMBL4829 O00763 Acetyl-CoA carboxylase 2 84.28% 98.00%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 83.05% 94.00%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 82.23% 99.23%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 82.21% 82.69%
CHEMBL3192 Q9BY41 Histone deacetylase 8 81.73% 93.99%
CHEMBL2708 Q16584 Mitogen-activated protein kinase kinase kinase 11 81.52% 81.14%
CHEMBL213 P08588 Beta-1 adrenergic receptor 81.50% 95.56%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 80.45% 85.00%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 80.22% 97.14%
CHEMBL2553 Q15418 Ribosomal protein S6 kinase alpha 1 80.05% 85.11%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 10030285
LOTUS LTS0087473
wikiData Q77573361