alpha-Cyclopiazonic acid

Details

Top
Internal ID 6173d372-d236-4466-bf3b-20230587470c
Taxonomy Organoheterocyclic compounds > Indoles and derivatives > Indoles > 3-alkylindoles
IUPAC Name (2R,3S,5Z,9R)-5-(1-hydroxyethylidene)-8,8-dimethyl-7,16-diazapentacyclo[9.6.1.02,9.03,7.015,18]octadeca-1(17),11(18),12,14-tetraene-4,6-dione
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C20H20N2O3/c1-9(23)14-18(24)17-16-11-8-21-13-6-4-5-10(15(11)13)7-12(16)20(2,3)22(17)19(14)25/h4-6,8,12,16-17,21,23H,7H2,1-3H3/b14-9-/t12-,16+,17+/m1/s1
InChI Key CNZIQHGDUXRUJS-PTNHGACKSA-N
Popularity 29 references in papers

Physical and Chemical Properties

Top
Molecular Formula C20H20N2O3
Molecular Weight 336.40 g/mol
Exact Mass 336.14739250 g/mol
Topological Polar Surface Area (TPSA) 73.40 Ų
XlogP 2.90

Synonyms

Top
CHEBI:22450
alpha-Cyclopiazonic acid
CHEMBL468766
83136-88-3
MFCD00167445
Cyclopiazonic acid from Penicillium cyclopium
Cyclopiazonic acid, 98%
(6aR,10Z,11aS,11bR)-10-(1-hydroxyethylidene)-7,7-dimethyl-6a,7,11a,11b-tetrahydro-6H-pyrrolo[1',2':2,3]isoindolo[4,5,6-cd]indole-9,11(2H,10H)-dione
CHEMBL480627
HMS1791B05
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

Top
2D Structure of alpha-Cyclopiazonic acid

3D Structure

Top

ADMET Properties (via admetSAR 2)

Top
Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

Top

Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
CHEMBL3901 P16615 Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 90 nM
IC50
via Super-PRED
CHEMBL2401 Q93084 Sarcoplasmic/endoplasmic reticulum calcium ATPase 3 90 nM
IC50
via Super-PRED

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.38% 96.09%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 97.19% 94.45%
CHEMBL2581 P07339 Cathepsin D 96.04% 98.95%
CHEMBL217 P14416 Dopamine D2 receptor 95.93% 95.62%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 95.14% 85.14%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.13% 91.11%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.47% 95.56%
CHEMBL2095226 P05556 Integrin alpha-5/beta-1 91.25% 96.39%
CHEMBL3137262 O60341 LSD1/CoREST complex 90.40% 97.09%
CHEMBL253 P34972 Cannabinoid CB2 receptor 90.29% 97.25%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 90.01% 93.03%
CHEMBL3192 Q9BY41 Histone deacetylase 8 87.45% 93.99%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 86.93% 93.40%
CHEMBL1293249 Q13887 Kruppel-like factor 5 85.79% 86.33%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 85.54% 99.23%
CHEMBL1994 P08235 Mineralocorticoid receptor 84.48% 100.00%
CHEMBL3310 Q96DB2 Histone deacetylase 11 82.81% 88.56%
CHEMBL5608 Q16288 NT-3 growth factor receptor 82.66% 95.89%
CHEMBL1902 P62942 FK506-binding protein 1A 82.51% 97.05%
CHEMBL1806 P11388 DNA topoisomerase II alpha 82.43% 89.00%
CHEMBL2553 Q15418 Ribosomal protein S6 kinase alpha 1 80.11% 85.11%

Plants that contains it

Top
Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
There are no matching plants.

Cross-Links

Top
PubChem 135494311
LOTUS LTS0179745
wikiData Q27102566