(Dha7)MC-RR

Details

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Internal ID 7f9cede7-5da1-4f28-94fa-504db743f4d7
Taxonomy Organic acids and derivatives > Peptidomimetics > Hybrid peptides
IUPAC Name (5R,8S,11R,12S,15S,18S,19S,22R)-8,15-bis[3-(diaminomethylideneamino)propyl]-18-[(1E,3E,5S,6S)-6-methoxy-3,5-dimethyl-7-phenylhepta-1,3-dienyl]-5,12,19-trimethyl-2-methylidene-3,6,9,13,16,20,25-heptaoxo-1,4,7,10,14,17,21-heptazacyclopentacosane-11,22-dicarboxylic acid
SMILES (Canonical) CC1C(NC(=O)C(NC(=O)C(C(NC(=O)C(NC(=O)C(NC(=O)C(=C)NC(=O)CCC(NC1=O)C(=O)O)C)CCCN=C(N)N)C(=O)O)C)CCCN=C(N)N)C=CC(=CC(C)C(CC2=CC=CC=C2)OC)C
SMILES (Isomeric) C[C@H]1[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)C(=C)NC(=O)CC[C@@H](NC1=O)C(=O)O)C)CCCN=C(N)N)C(=O)O)C)CCCN=C(N)N)/C=C/C(=C/[C@H](C)[C@H](CC2=CC=CC=C2)OC)/C
InChI InChI=1S/C48H73N13O12/c1-25(23-26(2)36(73-7)24-31-13-9-8-10-14-31)17-18-32-27(3)39(63)60-35(45(69)70)19-20-37(62)55-29(5)41(65)56-30(6)42(66)59-34(16-12-22-54-48(51)52)44(68)61-38(46(71)72)28(4)40(64)58-33(43(67)57-32)15-11-21-53-47(49)50/h8-10,13-14,17-18,23,26-28,30,32-36,38H,5,11-12,15-16,19-22,24H2,1-4,6-7H3,(H,55,62)(H,56,65)(H,57,67)(H,58,64)(H,59,66)(H,60,63)(H,61,68)(H,69,70)(H,71,72)(H4,49,50,53)(H4,51,52,54)/b18-17+,25-23+/t26-,27-,28-,30+,32-,33-,34-,35+,36-,38+/m0/s1
InChI Key ANEDRERLGQEWQI-UAWDZTONSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C48H73N13O12
Molecular Weight 1024.20 g/mol
Exact Mass 1023.55016481 g/mol
Topological Polar Surface Area (TPSA) 416.00 Ų
XlogP -0.40

Synonyms

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[Dha7]MC-RR
131022-02-1
7-Demethylmicrocystin RR
7-Desmethyl-microcystin-RR
DTXSID101046040
(5R,8S,11R,12S,15S,18S,19S,22R)-8,15-bis[3-(diaminomethylideneamino)propyl]-18-[(1E,3E,5S,6S)-6-methoxy-3,5-dimethyl-7-phenylhepta-1,3-dienyl]-5,12,19-trimethyl-2-methylidene-3,6,9,13,16,20,25-heptaoxo-1,4,7,10,14,17,21-heptazacyclopentacosane-11,22-dicarboxylic acid
Cyanoginosin LA, 1-(2,3-didehydroalanine)-3-L-arginine-5-L-arginine-

2D Structure

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2D Structure of (Dha7)MC-RR

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL4040 P28482 MAP kinase ERK2 99.58% 83.82%
CHEMBL2581 P07339 Cathepsin D 99.33% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.23% 96.09%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.42% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 97.41% 94.45%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.26% 95.56%
CHEMBL1293249 Q13887 Kruppel-like factor 5 92.52% 86.33%
CHEMBL5608 Q16288 NT-3 growth factor receptor 92.05% 95.89%
CHEMBL2288 Q13526 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 91.85% 91.71%
CHEMBL3137262 O60341 LSD1/CoREST complex 91.60% 97.09%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 91.27% 97.64%
CHEMBL3060 Q9Y345 Glycine transporter 2 91.15% 99.17%
CHEMBL1255126 O15151 Protein Mdm4 88.94% 90.20%
CHEMBL3837 P07711 Cathepsin L 88.07% 96.61%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 87.78% 95.50%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 87.48% 96.47%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 86.11% 95.89%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 85.74% 90.71%
CHEMBL4072 P07858 Cathepsin B 83.46% 93.67%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 83.06% 93.00%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 82.34% 92.88%
CHEMBL1937 Q92769 Histone deacetylase 2 82.21% 94.75%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 81.54% 100.00%
CHEMBL221 P23219 Cyclooxygenase-1 81.42% 90.17%
CHEMBL2959 Q08881 Tyrosine-protein kinase ITK/TSK 81.20% 95.00%
CHEMBL2535 P11166 Glucose transporter 81.12% 98.75%
CHEMBL5103 Q969S8 Histone deacetylase 10 81.08% 90.08%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 80.36% 93.03%
CHEMBL340 P08684 Cytochrome P450 3A4 80.36% 91.19%
CHEMBL2179 P04062 Beta-glucocerebrosidase 80.01% 85.31%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 6441234
LOTUS LTS0086021
wikiData Q104246641