YM-266183

Details

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Internal ID f054e3ec-6472-41d1-94a9-bf594d6fed64
Taxonomy Phenylpropanoids and polyketides > Macrolactams
IUPAC Name 2-[2-[(26Z)-26-ethylidene-12,29-bis(1-hydroxyethyl)-19-(2-hydroxypropan-2-yl)-14,21,28,31-tetraoxo-10,17,24,34-tetrathia-6,13,20,27,30,35,36,37,38-nonazahexacyclo[30.2.1.18,11.115,18.122,25.02,7]octatriaconta-1(35),2(7),3,5,8,11(38),15,18(37),22,25(36),32-undecaen-5-yl]-1,3-thiazol-4-yl]-N-[(E)-1-oxo-1-(2-oxopropylamino)but-2-en-2-yl]-1,3-thiazole-4-carboxamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C48H47N13O10S6/c1-8-23(36(65)49-12-19(3)62)51-37(66)27-15-74-45(56-27)31-18-75-44(58-31)25-11-10-22-34(50-25)26-13-76-46(53-26)33(21(5)64)60-39(68)29-17-77-47(57-29)35(48(6,7)71)61-40(69)30-16-73-43(55-30)24(9-2)52-41(70)32(20(4)63)59-38(67)28-14-72-42(22)54-28/h8-11,13-18,20-21,32-33,35,63-64,71H,12H2,1-7H3,(H,49,65)(H,51,66)(H,52,70)(H,59,67)(H,60,68)(H,61,69)/b23-8+,24-9-
InChI Key QFPBQHRZGAWLEX-AUVWRIHKSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C48H47N13O10S6
Molecular Weight 1158.40 g/mol
Exact Mass 1157.18931179 g/mol
Topological Polar Surface Area (TPSA) 512.00 Ų
XlogP 3.20

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of YM-266183

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 98.60% 98.95%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 97.87% 93.03%
CHEMBL1293267 Q9HC97 G-protein coupled receptor 35 97.59% 89.34%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.12% 91.11%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 96.22% 96.09%
CHEMBL230 P35354 Cyclooxygenase-2 95.53% 89.63%
CHEMBL3267 P48736 PI3-kinase p110-gamma subunit 95.44% 95.71%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 92.67% 99.23%
CHEMBL3830 Q2M2I8 Adaptor-associated kinase 92.31% 83.10%
CHEMBL3401 O75469 Pregnane X receptor 91.70% 94.73%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 91.12% 94.45%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 90.63% 96.90%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 90.48% 92.88%
CHEMBL3384 Q16512 Protein kinase N1 90.26% 80.71%
CHEMBL221 P23219 Cyclooxygenase-1 89.77% 90.17%
CHEMBL2553 Q15418 Ribosomal protein S6 kinase alpha 1 89.50% 85.11%
CHEMBL255 P29275 Adenosine A2b receptor 88.95% 98.59%
CHEMBL1907602 P06493 Cyclin-dependent kinase 1/cyclin B1 87.88% 91.24%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 87.66% 85.14%
CHEMBL5600 P27448 Serine/threonine-protein kinase c-TAK1 87.25% 88.81%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 86.18% 94.00%
CHEMBL213 P08588 Beta-1 adrenergic receptor 86.02% 95.56%
CHEMBL3359 P21462 Formyl peptide receptor 1 85.27% 93.56%
CHEMBL3975 P09467 Fructose-1,6-bisphosphatase 85.05% 92.95%
CHEMBL253 P34972 Cannabinoid CB2 receptor 83.49% 97.25%
CHEMBL2094135 Q96BI3 Gamma-secretase 82.98% 98.05%
CHEMBL4578 Q14680 Maternal embryonic leucine zipper kinase 82.92% 81.58%
CHEMBL1937 Q92769 Histone deacetylase 2 82.81% 94.75%
CHEMBL1806 P11388 DNA topoisomerase II alpha 82.66% 89.00%
CHEMBL2095226 P05556 Integrin alpha-5/beta-1 81.77% 96.39%
CHEMBL2335 P42785 Lysosomal Pro-X carboxypeptidase 81.64% 100.00%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 81.58% 90.71%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 81.00% 96.67%
CHEMBL3038469 P24941 CDK2/Cyclin A 80.79% 91.38%
CHEMBL4227 P25090 Lipoxin A4 receptor 80.70% 100.00%
CHEMBL2563 Q9UQL6 Histone deacetylase 5 80.56% 89.67%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 101237083
LOTUS LTS0077360
wikiData Q103817117