Paliurine I

Details

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Internal ID 91d1ce57-d152-4bd4-931d-1e7fc938a486
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Oligopeptides
IUPAC Name (2S,3S)-N-[(2S)-1-[(3S,10S,13E)-10-benzyl-16-methoxy-8,11-dioxo-2-oxa-6,9,12-triazatricyclo[13.3.1.03,7]nonadeca-1(19),13,15,17-tetraen-6-yl]-4-methyl-1-oxopentan-2-yl]-3-methyl-2-(methylamino)pentanamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C36H49N5O6/c1-7-23(4)31(37-5)34(43)40-28(19-22(2)3)36(45)41-18-16-30-32(41)35(44)39-27(20-24-11-9-8-10-12-24)33(42)38-17-15-25-21-26(47-30)13-14-29(25)46-6/h8-15,17,21-23,27-28,30-32,37H,7,16,18-20H2,1-6H3,(H,38,42)(H,39,44)(H,40,43)/b17-15+/t23-,27-,28-,30-,31-,32?/m0/s1
InChI Key LLZKJMREUXHIRU-AGVBJAGVSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C36H49N5O6
Molecular Weight 647.80 g/mol
Exact Mass 647.36828430 g/mol
Topological Polar Surface Area (TPSA) 138.00 Ų
XlogP 4.80

Synonyms

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RefChem:928511
(2S,3S)-N-((2S)-1-((3S,10S,13E)-10-benzyl-16-methoxy-8,11-dioxo-2-oxa-6,9,12-triazatricyclo(13.3.1.03,7)nonadeca-1(19),13,15,17-tetraen-6-yl)-4-methyl-1-oxopentan-2-yl)-3-methyl-2-(methylamino)pentanamide
403842-58-0

2D Structure

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2D Structure of Paliurine I

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.66% 98.95%
CHEMBL3837 P07711 Cathepsin L 99.27% 96.61%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.01% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 98.55% 85.14%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 96.37% 97.14%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 94.90% 97.64%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 93.50% 95.56%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 93.25% 94.45%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 92.19% 98.33%
CHEMBL204 P00734 Thrombin 91.86% 96.01%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 91.42% 95.89%
CHEMBL3060 Q9Y345 Glycine transporter 2 91.00% 99.17%
CHEMBL4208 P20618 Proteasome component C5 90.24% 90.00%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.19% 95.89%
CHEMBL1255126 O15151 Protein Mdm4 86.57% 90.20%
CHEMBL2413 P32246 C-C chemokine receptor type 1 86.29% 89.50%
CHEMBL4588 P22894 Matrix metalloproteinase 8 85.74% 94.66%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 85.37% 93.03%
CHEMBL2535 P11166 Glucose transporter 85.12% 98.75%
CHEMBL3359 P21462 Formyl peptide receptor 1 85.04% 93.56%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 84.98% 91.11%
CHEMBL5028 O14672 ADAM10 84.57% 97.50%
CHEMBL1293249 Q13887 Kruppel-like factor 5 83.75% 86.33%
CHEMBL340 P08684 Cytochrome P450 3A4 83.02% 91.19%
CHEMBL3137262 O60341 LSD1/CoREST complex 81.98% 97.09%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 81.79% 90.71%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Paliurus ramosissimus

Cross-Links

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PubChem 101204324
LOTUS LTS0071388
wikiData Q105153802