(4S)-4,5-dihydro-4-hydroxygeldanamycin

Details

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Internal ID 202b0ad7-e0a7-48f6-aa55-730c188a8ccf
Taxonomy Phenylpropanoids and polyketides > Macrolactams
IUPAC Name [(4E,6S,8S,9S,10E,12S,13R,14S,16R)-6,13-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18-tetraen-9-yl] carbamate
SMILES (Canonical) CC1CC(C(C(C=C(C(C(CC(C=C(C(=O)NC2=CC(=O)C(=C(C1)C2=O)OC)C)O)OC)OC(=O)N)C)C)O)OC
SMILES (Isomeric) C[C@H]1C[C@@H]([C@@H]([C@H](/C=C(/[C@@H]([C@H](C[C@@H](/C=C(/C(=O)NC2=CC(=O)C(=C(C1)C2=O)OC)\C)O)OC)OC(=O)N)\C)C)O)OC
InChI InChI=1S/C29H42N2O10/c1-14-8-19-25(35)20(13-21(33)27(19)40-7)31-28(36)17(4)11-18(32)12-23(39-6)26(41-29(30)37)16(3)10-15(2)24(34)22(9-14)38-5/h10-11,13-15,18,22-24,26,32,34H,8-9,12H2,1-7H3,(H2,30,37)(H,31,36)/b16-10+,17-11+/t14-,15+,18-,22+,23+,24-,26+/m1/s1
InChI Key HNYXYDNFRIJYMY-HBDFPOJRSA-N
Popularity 1 reference in papers

Physical and Chemical Properties

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Molecular Formula C29H42N2O10
Molecular Weight 578.70 g/mol
Exact Mass 578.28394554 g/mol
Topological Polar Surface Area (TPSA) 184.00 Ų
XlogP 0.90

Synonyms

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((4E,6S,8S,9S,10E,12S,13R,14S,16R)-6,13-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo(16.3.1)docosa-1(21),4,10,18-tetraen-9-yl) carbamate
[(4E,6S,8S,9S,10E,12S,13R,14S,16R)-6,13-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18-tetraen-9-yl] carbamate
RefChem:69541
CHEMBL2087235
CHEBI:205230

2D Structure

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2D Structure of (4S)-4,5-dihydro-4-hydroxygeldanamycin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.09% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 98.91% 85.14%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.76% 91.11%
CHEMBL241 Q14432 Phosphodiesterase 3A 95.88% 92.94%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.76% 95.56%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 93.94% 96.77%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 93.84% 94.45%
CHEMBL3137262 O60341 LSD1/CoREST complex 93.71% 97.09%
CHEMBL2581 P07339 Cathepsin D 93.60% 98.95%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 89.43% 99.23%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 88.76% 93.03%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 87.05% 96.95%
CHEMBL215 P09917 Arachidonate 5-lipoxygenase 86.96% 92.68%
CHEMBL221 P23219 Cyclooxygenase-1 86.83% 90.17%
CHEMBL2535 P11166 Glucose transporter 86.27% 98.75%
CHEMBL5608 Q16288 NT-3 growth factor receptor 86.00% 95.89%
CHEMBL253 P34972 Cannabinoid CB2 receptor 85.80% 97.25%
CHEMBL1806 P11388 DNA topoisomerase II alpha 83.91% 89.00%
CHEMBL1293249 Q13887 Kruppel-like factor 5 83.25% 86.33%
CHEMBL3267 P48736 PI3-kinase p110-gamma subunit 82.28% 95.71%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 81.77% 91.07%
CHEMBL1994 P08235 Mineralocorticoid receptor 80.56% 100.00%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 80.37% 97.33%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 66553960
LOTUS LTS0208097
wikiData Q77422953