epi-Ivermectin B1a

Details

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Internal ID 312d3620-b6e1-4a01-bac8-4a8862642be5
Taxonomy Phenylpropanoids and polyketides > Macrolides and analogues > Milbemycins
IUPAC Name 6'-butan-2-yl-21,24-dihydroxy-12-[5-(5-hydroxy-4-methoxy-6-methyloxan-2-yl)oxy-4-methoxy-6-methyloxan-2-yl]oxy-5',11,13,22-tetramethylspiro[3,7,19-trioxatetracyclo[15.6.1.14,8.020,24]pentacosa-10,14,16,22-tetraene-6,2'-oxane]-2-one
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C48H74O14/c1-11-25(2)43-28(5)17-18-47(62-43)23-34-20-33(61-47)16-15-27(4)42(26(3)13-12-14-32-24-55-45-40(49)29(6)19-35(46(51)58-34)48(32,45)52)59-39-22-37(54-10)44(31(8)57-39)60-38-21-36(53-9)41(50)30(7)56-38/h12-15,19,25-26,28,30-31,33-45,49-50,52H,11,16-18,20-24H2,1-10H3
InChI Key AZSNMRSAGSSBNP-UHFFFAOYSA-N
Popularity 4 references in papers

Physical and Chemical Properties

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Molecular Formula C48H74O14
Molecular Weight 875.10 g/mol
Exact Mass 874.50785703 g/mol
Topological Polar Surface Area (TPSA) 170.00 Ų
XlogP 4.10

Synonyms

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70288-86-7
71827-03-7
FT-0601609

2D Structure

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2D Structure of epi-Ivermectin B1a

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
CHEMBL1293235 P02545 Prelamin-A/C 398.1 nM
Potency
via Super-PRED
CHEMBL2842 P42345 Serine/threonine-protein kinase mTOR 3.3 nM
Potency
via Super-PRED
CHEMBL1963 P16473 Thyroid stimulating hormone receptor 31.6 nM
Potency
via Super-PRED

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.11% 96.09%
CHEMBL253 P34972 Cannabinoid CB2 receptor 97.63% 97.25%
CHEMBL4303 P08238 Heat shock protein HSP 90-beta 96.72% 96.77%
CHEMBL3137262 O60341 LSD1/CoREST complex 94.12% 97.09%
CHEMBL4793 Q86TI2 Dipeptidyl peptidase IX 93.63% 96.95%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 93.44% 91.11%
CHEMBL226 P30542 Adenosine A1 receptor 92.12% 95.93%
CHEMBL1871 P10275 Androgen Receptor 92.06% 96.43%
CHEMBL1293249 Q13887 Kruppel-like factor 5 91.58% 86.33%
CHEMBL1994 P08235 Mineralocorticoid receptor 90.74% 100.00%
CHEMBL1806 P11388 DNA topoisomerase II alpha 90.07% 89.00%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 89.37% 94.45%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 88.90% 96.47%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 88.49% 96.38%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 87.86% 94.00%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 87.59% 96.00%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 87.56% 95.56%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 86.23% 97.14%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 86.13% 99.23%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 86.08% 92.62%
CHEMBL5608 Q16288 NT-3 growth factor receptor 84.29% 95.89%
CHEMBL2140 P48775 Tryptophan 2,3-dioxygenase 83.44% 98.46%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 83.09% 95.89%
CHEMBL4208 P20618 Proteasome component C5 82.95% 90.00%
CHEMBL255 P29275 Adenosine A2b receptor 81.10% 98.59%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 80.82% 97.33%
CHEMBL2581 P07339 Cathepsin D 80.78% 98.95%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 4330618
LOTUS LTS0054405
wikiData Q104921907