22-O-(N-Me-L-valyl)-21-epi-aflaquinolone B

Details

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Internal ID 1caee8ce-7006-43a4-bd55-9ceba7edafb7
Taxonomy Organoheterocyclic compounds > Quinolines and derivatives > Phenylquinolines
IUPAC Name [(1R,2R,4R)-4-[(E)-2-[(3S,4S)-4,5-dihydroxy-3-methoxy-2-oxo-4-phenyl-1,3-dihydroquinolin-6-yl]ethenyl]-2,4-dimethylcyclohexyl] (2S)-3-methyl-2-(methylamino)butanoate
SMILES (Canonical) CC1CC(CCC1OC(=O)C(C(C)C)NC)(C)C=CC2=C(C3=C(C=C2)NC(=O)C(C3(C4=CC=CC=C4)O)OC)O
SMILES (Isomeric) C[C@@H]1C[C@](CC[C@H]1OC(=O)[C@H](C(C)C)NC)(C)/C=C/C2=C(C3=C(C=C2)NC(=O)[C@H]([C@@]3(C4=CC=CC=C4)O)OC)O
InChI InChI=1S/C32H42N2O6/c1-19(2)26(33-5)30(37)40-24-15-17-31(4,18-20(24)3)16-14-21-12-13-23-25(27(21)35)32(38,22-10-8-7-9-11-22)28(39-6)29(36)34-23/h7-14,16,19-20,24,26,28,33,35,38H,15,17-18H2,1-6H3,(H,34,36)/b16-14+/t20-,24-,26+,28-,31-,32+/m1/s1
InChI Key HXDOHVMCRWLYFS-XCNYLRODSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C32H42N2O6
Molecular Weight 550.70 g/mol
Exact Mass 550.30428706 g/mol
Topological Polar Surface Area (TPSA) 117.00 Ų
XlogP 4.90

Synonyms

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22-O-(N-Me-L-valyl)-21-epi-aflaquinolone B

2D Structure

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2D Structure of 22-O-(N-Me-L-valyl)-21-epi-aflaquinolone B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 99.67% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 98.76% 94.45%
CHEMBL2581 P07339 Cathepsin D 97.42% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.22% 96.09%
CHEMBL2035 P08912 Muscarinic acetylcholine receptor M5 97.04% 94.62%
CHEMBL216 P11229 Muscarinic acetylcholine receptor M1 96.90% 94.23%
CHEMBL221 P23219 Cyclooxygenase-1 95.24% 90.17%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 95.03% 95.56%
CHEMBL1821 P08173 Muscarinic acetylcholine receptor M4 93.67% 94.08%
CHEMBL3137262 O60341 LSD1/CoREST complex 93.14% 97.09%
CHEMBL1937 Q92769 Histone deacetylase 2 91.40% 94.75%
CHEMBL1293249 Q13887 Kruppel-like factor 5 90.97% 86.33%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 90.65% 93.03%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 89.77% 92.88%
CHEMBL1075094 Q16236 Nuclear factor erythroid 2-related factor 2 89.50% 96.00%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.99% 95.89%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 88.98% 96.47%
CHEMBL5028 O14672 ADAM10 87.85% 97.50%
CHEMBL3091268 Q92753 Nuclear receptor ROR-beta 86.09% 95.50%
CHEMBL1841 P06241 Tyrosine-protein kinase FYN 85.61% 81.29%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 85.24% 91.07%
CHEMBL2959 Q08881 Tyrosine-protein kinase ITK/TSK 84.24% 95.00%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 83.71% 82.69%
CHEMBL340 P08684 Cytochrome P450 3A4 82.60% 91.19%
CHEMBL4224 P49759 Dual specificty protein kinase CLK1 81.26% 85.30%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 101893728
LOTUS LTS0169443
wikiData Q105034938