2-Phenylamino-1,4-naphthoquinone

Details

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Internal ID 4a26504f-5a6f-47f0-8d93-335fdad49508
Taxonomy Benzenoids > Naphthalenes > Naphthoquinones
IUPAC Name 2-anilinonaphthalene-1,4-dione
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C16H11NO2/c18-15-10-14(17-11-6-2-1-3-7-11)16(19)13-9-5-4-8-12(13)15/h1-10,17H
InChI Key OPECBHGHSFBITB-UHFFFAOYSA-N
Popularity 34 references in papers

Physical and Chemical Properties

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Molecular Formula C16H11NO2
Molecular Weight 249.26 g/mol
Exact Mass 249.078978594 g/mol
Topological Polar Surface Area (TPSA) 46.20 Ų
XlogP 2.80

Synonyms

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RefChem:465235
2-Anilino-1,4-naphthoquinone
6628-97-3
2-(phenylamino)naphthalene-1,4-dione
2-anilinonaphthalene-1,4-dione
MLS001048869
SMR000387072
2-Anilinonaphthoquinone
CCRIS 6674
NSC59789
There are more than 10 synonyms. If you wish to see them all click here.

2D Structure

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2D Structure of 2-Phenylamino-1,4-naphthoquinone

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
CHEMBL3577 P00352 Aldehyde dehydrogenase 1A1 39810.7 nM
Potency
via CMAUP
CHEMBL5514 P42858 Huntingtin 11220.2 nM
Potency
via CMAUP
CHEMBL1287622 Q9Y468 Lethal(3)malignant brain tumor-like protein 1 2511.9 nM
Potency
via CMAUP
CHEMBL4040 P28482 MAP kinase ERK2 25118.9 nM
Potency
via CMAUP
CHEMBL1293224 P10636 Microtubule-associated protein tau 7079.5 nM
Potency
via CMAUP
CHEMBL1293277 O15118 Niemann-Pick C1 protein 1778.3 nM
Potency
via CMAUP
CHEMBL1293235 P02545 Prelamin-A/C 17.8 nM
17.8 nM
Potency
Potency
via Super-PRED
via CMAUP
CHEMBL1293294 P51151 Ras-related protein Rab-9A 1000 nM
Potency
via CMAUP
CHEMBL1293232 Q16637 Survival motor neuron protein 12589.3 nM
Potency
via CMAUP

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 96.15% 95.56%
CHEMBL2581 P07339 Cathepsin D 91.83% 98.95%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 90.39% 96.67%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 90.07% 82.69%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 89.28% 99.23%
CHEMBL221 P23219 Cyclooxygenase-1 87.16% 90.17%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 84.99% 93.03%
CHEMBL216 P11229 Muscarinic acetylcholine receptor M1 83.07% 94.23%
CHEMBL2535 P11166 Glucose transporter 81.99% 98.75%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
To see more specific details click the taxa you are interested in.
Lygodium japonicum

Cross-Links

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PubChem 81124
NPASS NPC192533
ChEMBL CHEMBL84010