Sch 20562

Details

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Internal ID 4c0eb3d5-6f56-477a-9a32-da1d3eda0074
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides > Cyclic glycodepsipeptides
IUPAC Name (3R)-N-[(E)-1-[[(3S,6S,12R,15E,18R,21R,24S,25R)-12-(3-amino-3-oxopropyl)-15-ethylidene-21-[(1R)-1-hydroxyethyl]-18-[(4-hydroxyphenyl)methyl]-3-(1H-imidazol-5-ylmethyl)-7,25-dimethyl-2,5,8,11,14,17,20,23-octaoxo-6-[(1S)-1-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyethyl]-1-oxa-4,7,10,13,16,19,22-heptazacyclopentacos-24-yl]amino]-1-oxobut-2-en-2-yl]-3-hydroxytetradecanamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C63H96N12O21/c1-8-11-12-13-14-15-16-17-18-19-39(79)28-47(81)68-40(9-2)57(88)74-50-34(5)94-62(93)44(27-37-29-65-32-67-37)72-61(92)51(35(6)95-63-54(85)53(84)52(83)45(31-76)96-63)75(7)48(82)30-66-55(86)42(24-25-46(64)80)70-56(87)41(10-3)69-58(89)43(26-36-20-22-38(78)23-21-36)71-59(90)49(33(4)77)73-60(50)91/h9-10,20-23,29,32-35,39,42-45,49-54,63,76-79,83-85H,8,11-19,24-28,30-31H2,1-7H3,(H2,64,80)(H,65,67)(H,66,86)(H,68,81)(H,69,89)(H,70,87)(H,71,90)(H,72,92)(H,73,91)(H,74,88)/b40-9+,41-10+/t33-,34-,35+,39-,42-,43-,44+,45-,49-,50+,51+,52-,53+,54-,63+/m1/s1
InChI Key JZKVLKBVTSOCID-NJJAETPXSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C63H96N12O21
Molecular Weight 1357.50 g/mol
Exact Mass 1356.68129812 g/mol
Topological Polar Surface Area (TPSA) 511.00 Ų
XlogP 0.80

Synonyms

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Sch-20562
RefChem:181719
69856-27-5
CHEBI:218650

2D Structure

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2D Structure of Sch 20562

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 99.75% 96.09%
CHEMBL2581 P07339 Cathepsin D 99.44% 98.95%
CHEMBL3038469 P24941 CDK2/Cyclin A 99.19% 91.38%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.89% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 97.84% 94.45%
CHEMBL2107 P61073 C-X-C chemokine receptor type 4 97.35% 93.10%
CHEMBL3060 Q9Y345 Glycine transporter 2 97.30% 99.17%
CHEMBL5103 Q969S8 Histone deacetylase 10 96.51% 90.08%
CHEMBL4040 P28482 MAP kinase ERK2 95.89% 83.82%
CHEMBL5608 Q16288 NT-3 growth factor receptor 94.95% 95.89%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 94.69% 100.00%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 94.64% 97.33%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 94.12% 96.90%
CHEMBL2996 Q05655 Protein kinase C delta 93.84% 97.79%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 93.42% 97.64%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 93.19% 85.14%
CHEMBL2955 O95136 Sphingosine 1-phosphate receptor Edg-5 92.28% 92.86%
CHEMBL1907605 P24864 Cyclin-dependent kinase 2/cyclin E1 90.56% 92.88%
CHEMBL2208 P49137 MAP kinase-activated protein kinase 2 90.16% 95.20%
CHEMBL1907602 P06493 Cyclin-dependent kinase 1/cyclin B1 89.77% 91.24%
CHEMBL1806 P11388 DNA topoisomerase II alpha 89.69% 89.00%
CHEMBL255 P29275 Adenosine A2b receptor 89.30% 98.59%
CHEMBL3137262 O60341 LSD1/CoREST complex 89.23% 97.09%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 89.02% 85.00%
CHEMBL2514 O95665 Neurotensin receptor 2 88.65% 100.00%
CHEMBL4588 P22894 Matrix metalloproteinase 8 88.56% 94.66%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 88.29% 90.71%
CHEMBL226 P30542 Adenosine A1 receptor 88.02% 95.93%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 87.86% 95.89%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 87.85% 82.38%
CHEMBL253 P34972 Cannabinoid CB2 receptor 87.65% 97.25%
CHEMBL2563 Q9UQL6 Histone deacetylase 5 87.04% 89.67%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 86.46% 99.23%
CHEMBL4227 P25090 Lipoxin A4 receptor 86.27% 100.00%
CHEMBL2535 P11166 Glucose transporter 85.26% 98.75%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 85.16% 95.56%
CHEMBL3359 P21462 Formyl peptide receptor 1 84.61% 93.56%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 84.54% 93.00%
CHEMBL5469 Q14289 Protein tyrosine kinase 2 beta 83.89% 91.03%
CHEMBL3891 P07384 Calpain 1 83.57% 93.04%
CHEMBL2096618 P11274 Bcr/Abl fusion protein 83.55% 85.83%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 83.54% 95.50%
CHEMBL1937 Q92769 Histone deacetylase 2 83.37% 94.75%
CHEMBL5555 O00767 Acyl-CoA desaturase 83.23% 97.50%
CHEMBL221 P23219 Cyclooxygenase-1 82.82% 90.17%
CHEMBL5043 Q6P179 Endoplasmic reticulum aminopeptidase 2 82.51% 91.81%
CHEMBL1293249 Q13887 Kruppel-like factor 5 81.88% 86.33%
CHEMBL3476 O15111 Inhibitor of nuclear factor kappa B kinase alpha subunit 81.21% 95.83%
CHEMBL3401 O75469 Pregnane X receptor 80.97% 94.73%
CHEMBL2635 P51452 Dual specificity protein phosphatase 3 80.71% 94.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 10796528
LOTUS LTS0070128
wikiData Q77502029