11,12-Epoxypukalide

Details

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Internal ID d9a62b48-d90e-4f18-8604-e285d5d397cd
Taxonomy Phenylpropanoids and polyketides > Macrolides and analogues
IUPAC Name methyl (1R,4S,10R,12S,14R,15R)-12-methyl-17-oxo-4-prop-1-en-2-yl-11,16,18,19-tetraoxapentacyclo[12.2.2.16,9.01,15.010,12]nonadeca-6,8-diene-7-carboxylate
SMILES (Canonical) CC(=C)C1CCC23C(O2)C(CC4(C(O4)C5=CC(=C(C1)O5)C(=O)OC)C)OC3=O
SMILES (Isomeric) CC(=C)[C@H]1CC[C@]23[C@H](O2)[C@@H](C[C@]4([C@@H](O4)C5=CC(=C(C1)O5)C(=O)OC)C)OC3=O
InChI InChI=1S/C21H24O7/c1-10(2)11-5-6-21-17(28-21)15(26-19(21)23)9-20(3)16(27-20)14-8-12(18(22)24-4)13(7-11)25-14/h8,11,15-17H,1,5-7,9H2,2-4H3/t11-,15+,16-,17+,20-,21+/m0/s1
InChI Key QKPWPHBMPBPNMQ-FELIULDUSA-N
Popularity 3 references in papers

Physical and Chemical Properties

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Molecular Formula C21H24O7
Molecular Weight 388.40 g/mol
Exact Mass 388.15220310 g/mol
Topological Polar Surface Area (TPSA) 90.80 Ų
XlogP 2.60

Synonyms

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95925-22-7
methyl (1R,4S,10R,12S,14R,15R)-12-methyl-17-oxo-4-prop-1-en-2-yl-11,16,18,19-tetraoxapentacyclo[12.2.2.16,9.01,15.010,12]nonadeca-6,8-diene-7-carboxylate
SCHEMBL2317764
DTXSID20914736
11,16,18,19-Tetraoxapentacyclo(12.2.2.1(6,9).0(1,15).0(10,12))nonadeca-6,8-diene-7-carboxylic acid, 12-methyl-4-(1-methylethenyl)-17-oxo-, methyl ester, (1R-(1R*,4S*,10R*,12S*,14R*,15R*))-
Methyl 12-methyl-17-oxo-4-(prop-1-en-2-yl)-11,16,18,19-tetraoxapentacyclo[12.2.2.1~6,9~.0~1,15~.0~10,12~]nonadeca-6,8-diene-7-carboxylate

2D Structure

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2D Structure of 11,12-Epoxypukalide

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 98.36% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 95.76% 94.45%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 94.62% 96.09%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 90.96% 85.14%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.07% 95.89%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 87.71% 97.14%
CHEMBL1293249 Q13887 Kruppel-like factor 5 87.62% 86.33%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 87.30% 93.03%
CHEMBL3713062 P10646 Tissue factor pathway inhibitor 86.73% 97.33%
CHEMBL340 P08684 Cytochrome P450 3A4 86.00% 91.19%
CHEMBL1907602 P06493 Cyclin-dependent kinase 1/cyclin B1 84.54% 91.24%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 82.53% 96.90%
CHEMBL241 Q14432 Phosphodiesterase 3A 82.41% 92.94%
CHEMBL3137262 O60341 LSD1/CoREST complex 82.11% 97.09%
CHEMBL2007 P16234 Platelet-derived growth factor receptor alpha 82.03% 91.07%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 81.72% 92.62%
CHEMBL4051 P13569 Cystic fibrosis transmembrane conductance regulator 80.92% 95.71%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 146895
LOTUS LTS0081723
wikiData Q82885551