11-Acetoxy-N-hydroxymethyl-pretubulysin

Details

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Internal ID 6932a211-e0e7-48f7-8a1d-8c4d9992d48b
Taxonomy Organic acids and derivatives > Carboxylic acids and derivatives > Amino acids, peptides, and analogues > Peptides > Dipeptides
IUPAC Name (2S,4R)-4-[[2-[(3R)-1-acetyloxy-3-[hydroxymethyl-[(2S,3S)-3-methyl-2-[[(2R)-1-methylpiperidine-2-carbonyl]amino]pentanoyl]amino]-4-methylpentyl]-1,3-thiazole-4-carbonyl]amino]-2-methyl-5-phenylpentanoic acid
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C38H57N5O8S/c1-8-24(4)33(41-35(47)30-16-12-13-17-42(30)7)37(48)43(22-44)31(23(2)3)20-32(51-26(6)45)36-40-29(21-52-36)34(46)39-28(18-25(5)38(49)50)19-27-14-10-9-11-15-27/h9-11,14-15,21,23-25,28,30-33,44H,8,12-13,16-20,22H2,1-7H3,(H,39,46)(H,41,47)(H,49,50)/t24-,25-,28+,30+,31+,32?,33-/m0/s1
InChI Key IVAMWOWNWPBUJU-ZTJQOVPWSA-N
Popularity 2 references in papers

Physical and Chemical Properties

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Molecular Formula C38H57N5O8S
Molecular Weight 744.00 g/mol
Exact Mass 743.39278497 g/mol
Topological Polar Surface Area (TPSA) 207.00 Ų
XlogP 3.20

Synonyms

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There are no found synonyms.

2D Structure

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2D Structure of 11-Acetoxy-N-hydroxymethyl-pretubulysin

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.88% 98.95%
CHEMBL4072 P07858 Cathepsin B 98.70% 93.67%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.55% 96.09%
CHEMBL221 P23219 Cyclooxygenase-1 97.29% 90.17%
CHEMBL1795139 Q8IU80 Transmembrane protease serine 6 94.66% 98.33%
CHEMBL253 P34972 Cannabinoid CB2 receptor 92.46% 97.25%
CHEMBL3359 P21462 Formyl peptide receptor 1 92.27% 93.56%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 91.13% 97.64%
CHEMBL240 Q12809 HERG 90.73% 89.76%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 90.21% 95.56%
CHEMBL340 P08684 Cytochrome P450 3A4 89.87% 91.19%
CHEMBL226 P30542 Adenosine A1 receptor 89.59% 95.93%
CHEMBL3837 P07711 Cathepsin L 89.55% 96.61%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 89.00% 93.00%
CHEMBL235 P37231 Peroxisome proliferator-activated receptor gamma 84.35% 95.39%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 83.79% 99.23%
CHEMBL4227 P25090 Lipoxin A4 receptor 82.42% 100.00%
CHEMBL1741221 Q9Y4P1 Cysteine protease ATG4B 82.37% 87.50%
CHEMBL4208 P20618 Proteasome component C5 82.06% 90.00%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 81.58% 85.14%
CHEMBL2373 P21730 C5a anaphylatoxin chemotactic receptor 81.41% 92.62%
CHEMBL5028 O14672 ADAM10 81.34% 97.50%
CHEMBL3024 P53350 Serine/threonine-protein kinase PLK1 81.29% 97.43%
CHEMBL3430907 Q96GD4 Aurora kinase B/Inner centromere protein 80.48% 97.50%
CHEMBL5608 Q16288 NT-3 growth factor receptor 80.47% 95.89%
CHEMBL3060 Q9Y345 Glycine transporter 2 80.13% 99.17%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 139586394
LOTUS LTS0204292
wikiData Q77505520