(+)-3,4-dihydro-3,8-dihydroxy-3-methylbenz(a)anthracene-1,7,12(2H)-trione

Details

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Internal ID 643cb410-ddbc-4860-8ac1-48932832fec6
Taxonomy Phenylpropanoids and polyketides > Angucyclines
IUPAC Name (3R)-3,8-dihydroxy-3-methyl-2,4-dihydrobenzo[a]anthracene-1,7,12-trione
SMILES (Canonical) CC1(CC2=C(C(=O)C1)C3=C(C=C2)C(=O)C4=C(C3=O)C=CC=C4O)O
SMILES (Isomeric) C[C@]1(CC2=C(C(=O)C1)C3=C(C=C2)C(=O)C4=C(C3=O)C=CC=C4O)O
InChI InChI=1S/C19H14O5/c1-19(24)7-9-5-6-11-16(14(9)13(21)8-19)18(23)10-3-2-4-12(20)15(10)17(11)22/h2-6,20,24H,7-8H2,1H3/t19-/m1/s1
InChI Key UGEKKXLEYACFTD-LJQANCHMSA-N
Popularity 27 references in papers

Physical and Chemical Properties

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Molecular Formula C19H14O5
Molecular Weight 322.30 g/mol
Exact Mass 322.08412354 g/mol
Topological Polar Surface Area (TPSA) 91.70 Ų
XlogP 2.40

Synonyms

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(-)-tetrangomycin
CHEBI:32211
(3R)-3,8-dihydroxy-3-methyl-3,4-dihydrotetraphene-1,7,12(2H)-trione
(+)-3,4-dihydro-3,8-dihydroxy-3-methylbenz(a)anthracene- 1,7,12(2H)-trione
CHEMBL1668772
(+)-3,4-Dihydro-3,8-dihydroxy-3-methylbenz(a)anthracene-1,7,12(2H)-trione
Q27114829
(3R)-3,8-dihydroxy-3-methyl-2,4-dihydrobenzo[a]anthracene-1,7,12-trione

2D Structure

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2D Structure of (+)-3,4-dihydro-3,8-dihydroxy-3-methylbenz(a)anthracene-1,7,12(2H)-trione

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 98.07% 98.95%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 97.23% 91.11%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 96.54% 95.56%
CHEMBL1951 P21397 Monoamine oxidase A 95.50% 91.49%
CHEMBL1937 Q92769 Histone deacetylase 2 93.94% 94.75%
CHEMBL3038477 P67870 Casein kinase II alpha/beta 91.24% 99.23%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 91.16% 93.03%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 88.69% 96.09%
CHEMBL4026 P40763 Signal transducer and activator of transcription 3 87.46% 82.69%
CHEMBL2378 P30307 Dual specificity phosphatase Cdc25C 86.55% 96.67%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 85.70% 96.38%
CHEMBL1293249 Q13887 Kruppel-like factor 5 83.68% 86.33%
CHEMBL3492 P49721 Proteasome Macropain subunit 83.48% 90.24%
CHEMBL1806 P11388 DNA topoisomerase II alpha 83.21% 89.00%
CHEMBL1860 P10827 Thyroid hormone receptor alpha 82.12% 99.15%
CHEMBL240 Q12809 HERG 81.83% 89.76%
CHEMBL1994 P08235 Mineralocorticoid receptor 81.78% 100.00%
CHEMBL5697 Q9GZT9 Egl nine homolog 1 80.45% 93.40%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 11738774
LOTUS LTS0084873
wikiData Q27114829