Veraguamide B

Details

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Internal ID 7647f87a-c389-4b39-a6ac-1a3883a7b7d3
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name (3S,6S,9S,12S,13R,16S,19S)-13-(5-bromopent-4-ynyl)-7,12,17-trimethyl-3,6,9,16-tetra(propan-2-yl)-4,14-dioxa-1,7,10,17-tetrazabicyclo[17.3.0]docosane-2,5,8,11,15,18-hexone
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C36H57BrN4O8/c1-20(2)27-33(44)40(11)29(22(5)6)36(47)49-30(23(7)8)34(45)41-19-15-16-25(41)32(43)39(10)28(21(3)4)35(46)48-26(17-13-12-14-18-37)24(9)31(42)38-27/h20-30H,12-13,15-17,19H2,1-11H3,(H,38,42)/t24-,25-,26+,27-,28-,29-,30-/m0/s1
InChI Key UQYHDSHIIDYSSP-PYYGQVSISA-N
Popularity 5 references in papers

Physical and Chemical Properties

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Molecular Formula C36H57BrN4O8
Molecular Weight 753.80 g/mol
Exact Mass 752.33598 g/mol
Topological Polar Surface Area (TPSA) 143.00 Ų
XlogP 6.60

Synonyms

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(3S,6R,7S,10S,13S,16S,21aS)-6-(5-bromopent-4-yn-1-yl)-3,10,13,16-tetraisopropyl-2,7,12-trimethyldecahydro-6H-pyrrolo(2,1-f)(1,10)dioxa(4,7,13,16)tetraazacyclononadecine-1,4,8,11,14,17(7H,16H)-hexaone
(3S,6R,7S,10S,13S,16S,21aS)-6-(5-bromopent-4-yn-1-yl)-3,10,13,16-tetraisopropyl-2,7,12-trimethyldecahydro-6H-pyrrolo[2,1-f][1,10]dioxa[4,7,13,16]tetraazacyclononadecine-1,4,8,11,14,17(7H,16H)-hexaone
(3S,6S,9S,12S,13R,16S,19S)-13-(5-bromopent-4-ynyl)-7,12,17-trimethyl-3,6,9,16-tetra(propan-2-yl)-4,14-dioxa-1,7,10,17-tetrazabicyclo(17.3.0)docosane-2,5,8,11,15,18-hexone
(3S,6S,9S,12S,13R,16S,19S)-13-(5-bromopent-4-ynyl)-7,12,17-trimethyl-3,6,9,16-tetra(propan-2-yl)-4,14-dioxa-1,7,10,17-tetrazabicyclo[17.3.0]docosane-2,5,8,11,15,18-hexone
RefChem:193944
CHEMBL1783106
SCHEMBL29885818
CHEBI:67331
DTXSID201334767
Q27135788

2D Structure

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2D Structure of Veraguamide B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.15% 98.95%
CHEMBL333 P08253 Matrix metalloproteinase-2 98.78% 96.31%
CHEMBL5103 Q969S8 Histone deacetylase 10 98.26% 90.08%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 97.59% 96.09%
CHEMBL253 P34972 Cannabinoid CB2 receptor 96.65% 97.25%
CHEMBL4588 P22894 Matrix metalloproteinase 8 96.26% 94.66%
CHEMBL5203 P33316 dUTP pyrophosphatase 96.14% 99.18%
CHEMBL1978 P11511 Cytochrome P450 19A1 94.90% 91.76%
CHEMBL3837 P07711 Cathepsin L 94.79% 96.61%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 94.72% 95.56%
CHEMBL228 P31645 Serotonin transporter 92.53% 95.51%
CHEMBL2069156 Q14145 Kelch-like ECH-associated protein 1 91.81% 82.38%
CHEMBL321 P14780 Matrix metalloproteinase 9 91.28% 92.12%
CHEMBL4261 Q16665 Hypoxia-inducible factor 1 alpha 90.68% 85.14%
CHEMBL1902 P62942 FK506-binding protein 1A 89.63% 97.05%
CHEMBL3137262 O60341 LSD1/CoREST complex 89.25% 97.09%
CHEMBL1937 Q92769 Histone deacetylase 2 89.00% 94.75%
CHEMBL5608 Q16288 NT-3 growth factor receptor 88.98% 95.89%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 88.97% 90.71%
CHEMBL255 P29275 Adenosine A2b receptor 87.60% 98.59%
CHEMBL3310 Q96DB2 Histone deacetylase 11 86.01% 88.56%
CHEMBL1949 P62937 Cyclophilin A 85.82% 98.57%
CHEMBL3384 Q16512 Protein kinase N1 84.40% 80.71%
CHEMBL4187 Q99250 Sodium channel protein type II alpha subunit 84.33% 95.50%
CHEMBL6136 O60341 Lysine-specific histone demethylase 1 83.49% 95.58%
CHEMBL1871 P10275 Androgen Receptor 83.38% 96.43%
CHEMBL1907600 Q00535 Cyclin-dependent kinase 5/CDK5 activator 1 83.12% 93.03%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 82.38% 100.00%
CHEMBL2443 P49862 Kallikrein 7 82.35% 94.00%
CHEMBL1994 P08235 Mineralocorticoid receptor 82.31% 100.00%
CHEMBL325 Q13547 Histone deacetylase 1 82.03% 95.92%
CHEMBL2189110 Q15910 Histone-lysine N-methyltransferase EZH2 81.70% 97.50%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 81.55% 96.38%
CHEMBL332 P03956 Matrix metalloproteinase-1 81.03% 94.50%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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There are no matching plants.

Cross-Links

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PubChem 53355337
LOTUS LTS0020403
wikiData Q27135788