Aeruginopeptin 917S-B

Details

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Internal ID 0977d089-3c21-4153-b1a3-4adaa9a68767
Taxonomy Organic acids and derivatives > Peptidomimetics > Depsipeptides > Cyclic depsipeptides
IUPAC Name N-[8-butan-2-yl-21-hydroxy-15-[(4-hydroxycyclohex-2-en-1-yl)methyl]-5-[(4-hydroxyphenyl)methyl]-4,11-dimethyl-2-(2-methylpropyl)-3,6,9,13,16,22-hexaoxo-10-oxa-1,4,7,14,17-pentazabicyclo[16.3.1]docosan-12-yl]-2-[[2-hydroxy-3-(4-hydroxyphenyl)propanoyl]amino]pentanediamide
SMILES (Canonical)
SMILES (Isomeric)
InChI InChI=1S/C54H76N8O15/c1-7-29(4)45-54(76)77-30(5)46(60-47(69)37(20-22-43(55)67)56-50(72)42(66)27-33-12-18-36(65)19-13-33)51(73)58-39(25-31-8-14-34(63)15-9-31)48(70)57-38-21-23-44(68)62(52(38)74)41(24-28(2)3)53(75)61(6)40(49(71)59-45)26-32-10-16-35(64)17-11-32/h8,10-14,16-19,28-31,34,37-42,44-46,63-66,68H,7,9,15,20-27H2,1-6H3,(H2,55,67)(H,56,72)(H,57,70)(H,58,73)(H,59,71)(H,60,69)
InChI Key OZABBUPKYTXOSK-UHFFFAOYSA-N
Popularity 0 references in papers

Physical and Chemical Properties

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Molecular Formula C54H76N8O15
Molecular Weight 1077.20 g/mol
Exact Mass 1076.54301375 g/mol
Topological Polar Surface Area (TPSA) 357.00 Ų
XlogP 2.40

Synonyms

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CHEBI:80077
Q27149230
N-[8-butan-2-yl-21-hydroxy-15-[(4-hydroxycyclohex-2-en-1-yl)methyl]-5-[(4-hydroxyphenyl)methyl]-4,11-dimethyl-2-(2-methylpropyl)-3,6,9,13,16,22-hexaoxo-10-oxa-1,4,7,14,17-pentazabicyclo[16.3.1]docosan-12-yl]-2-[[2-hydroxy-3-(4-hydroxyphenyl)propanoyl]amino]pentanediamide

2D Structure

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2D Structure of Aeruginopeptin 917S-B

3D Structure

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ADMET Properties (via admetSAR 2)

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Target Value Probability (raw) Probability (%)
No predicted properties yet!

Targets

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Proven Targets:

CHEMBL ID UniProt ID Name Min activity Assay type Source
No proven targets yet!

Predicted Targets (via Super-PRED):

CHEMBL ID UniProt ID Name Probability Model accuracy
CHEMBL2581 P07339 Cathepsin D 99.85% 98.95%
CHEMBL3251 P19838 Nuclear factor NF-kappa-B p105 subunit 98.88% 96.09%
CHEMBL3837 P07711 Cathepsin L 97.46% 96.61%
CHEMBL4040 P28482 MAP kinase ERK2 97.16% 83.82%
CHEMBL2094135 Q96BI3 Gamma-secretase 96.45% 98.05%
CHEMBL221 P23219 Cyclooxygenase-1 96.38% 90.17%
CHEMBL3137262 O60341 LSD1/CoREST complex 95.65% 97.09%
CHEMBL5619 P27695 DNA-(apurinic or apyrimidinic site) lyase 94.73% 91.11%
CHEMBL4203 Q9HAZ1 Dual specificity protein kinase CLK4 94.67% 94.45%
CHEMBL3060 Q9Y345 Glycine transporter 2 93.37% 99.17%
CHEMBL3807 P17706 T-cell protein-tyrosine phosphatase 93.32% 93.00%
CHEMBL5103 Q969S8 Histone deacetylase 10 93.16% 90.08%
CHEMBL1907603 Q05586 Glutamate NMDA receptor; GRIN1/GRIN2B 93.08% 95.89%
CHEMBL3108638 O15164 Transcription intermediary factor 1-alpha 92.50% 95.56%
CHEMBL3359 P21462 Formyl peptide receptor 1 91.68% 93.56%
CHEMBL1806 P11388 DNA topoisomerase II alpha 90.96% 89.00%
CHEMBL2693 Q9UIQ6 Cystinyl aminopeptidase 90.89% 97.64%
CHEMBL236 P41143 Delta opioid receptor 90.66% 99.35%
CHEMBL5845 P23415 Glycine receptor subunit alpha-1 90.34% 90.71%
CHEMBL253 P34972 Cannabinoid CB2 receptor 90.05% 97.25%
CHEMBL5608 Q16288 NT-3 growth factor receptor 89.94% 95.89%
CHEMBL2000 P03952 Plasma kallikrein 89.43% 93.92%
CHEMBL1949 P62937 Cyclophilin A 88.84% 98.57%
CHEMBL4478 Q00975 Voltage-gated N-type calcium channel alpha-1B subunit 88.62% 97.14%
CHEMBL4588 P22894 Matrix metalloproteinase 8 88.57% 94.66%
CHEMBL2413 P32246 C-C chemokine receptor type 1 88.36% 89.50%
CHEMBL4227 P25090 Lipoxin A4 receptor 87.75% 100.00%
CHEMBL2514 O95665 Neurotensin receptor 2 87.53% 100.00%
CHEMBL333 P08253 Matrix metalloproteinase-2 86.02% 96.31%
CHEMBL3392948 Q9NP59 Solute carrier family 40 member 1 85.86% 95.00%
CHEMBL4685 P14902 Indoleamine 2,3-dioxygenase 85.14% 96.38%
CHEMBL4296 Q15858 Sodium channel protein type IX alpha subunit 85.13% 96.11%
CHEMBL255 P29275 Adenosine A2b receptor 82.99% 98.59%
CHEMBL2492 P36544 Neuronal acetylcholine receptor protein alpha-7 subunit 82.83% 88.42%
CHEMBL3130 O00329 PI3-kinase p110-delta subunit 82.75% 96.47%
CHEMBL1907594 P30926 Neuronal acetylcholine receptor; alpha3/beta4 81.89% 97.23%
CHEMBL2072 P35499 Sodium channel protein type IV alpha subunit 81.87% 92.32%
CHEMBL2111367 P27986 PI3-kinase p110-alpha/p85-alpha 81.71% 94.33%
CHEMBL340 P08684 Cytochrome P450 3A4 81.68% 91.19%
CHEMBL4072 P07858 Cathepsin B 81.55% 93.67%
CHEMBL5852 Q96P65 Pyroglutamylated RFamide peptide receptor 81.42% 85.00%
CHEMBL1075317 P61964 WD repeat-containing protein 5 81.20% 96.33%
CHEMBL3830 Q2M2I8 Adaptor-associated kinase 80.80% 83.10%
CHEMBL5163 Q9NY46 Sodium channel protein type III alpha subunit 80.78% 96.90%
CHEMBL2274 Q9H228 Sphingosine 1-phosphate receptor Edg-8 80.24% 100.00%

Plants that contains it

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Below are displayed all the plants proven (via scientific papers) to contain this compound!
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Cross-Links

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PubChem 23724564
LOTUS LTS0056488
wikiData Q27149230